Methods of using substituted isoxazolo pyridinones as dissociated glucocorticoids

A method for treating a subject having an inflammatory or auto-immune disease with a substituted isoxazolo pyridinone. Also, a method for administering a substituted isoxazolo pyridinone to a cell to retain or increase glucocorticoid receptor transrepression activity with only minimal glucocorticoid...

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Bibliographische Detailangaben
Hauptverfasser: Xu, Huaqiang Eric, Xu, Yong, He, Yuanzheng
Format: Patent
Sprache:eng
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Zusammenfassung:A method for treating a subject having an inflammatory or auto-immune disease with a substituted isoxazolo pyridinone. Also, a method for administering a substituted isoxazolo pyridinone to a cell to retain or increase glucocorticoid receptor transrepression activity with only minimal glucocorticoid receptor transactivation activity.