Method for producing quinolone carboxylic acid derivative

The present invention relates to a method for producing a quinolone compound having high antibacterial activity and high safety, at high yield and in a simple manner.A quinolonecarboxylic acid derivative (1) of interest is produced through a one-pot manner by reacting a compound (2) with a salt of a...

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Bibliographische Detailangaben
Hauptverfasser: Sato, Koji, Sakuratani, Kenji
Format: Patent
Sprache:eng
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Beschreibung
Zusammenfassung:The present invention relates to a method for producing a quinolone compound having high antibacterial activity and high safety, at high yield and in a simple manner.A quinolonecarboxylic acid derivative (1) of interest is produced through a one-pot manner by reacting a compound (2) with a salt of a cyclic amine (3) and with a boron derivative in a solvent in the presence of a base.