Process for the preparation of omega-benzyl esters of amino diacids and of alkanesulphonates of these esters, and these alkanesulphonates
The invention relates to a process for the preparation of an -benzyl ester of an amino diacid, characterized in that the amino diacid is reacted with a benzyl alcohol derivative of formula (I) 1 in which the R 1 substituent or substituents, which are identical or different, represent a hydrogen atom...
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Sprache: | eng |
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Zusammenfassung: | The invention relates to a process for the preparation of an -benzyl ester of an amino diacid, characterized in that the amino diacid is reacted with a benzyl alcohol derivative of formula (I)
1
in which the R
1
substituent or substituents, which are identical or different, represent a hydrogen atom, a C
1
to C
4
alkyl group, a C
1
to C
4
alkoxy group or a halogen atom and n is equal to 1, 2 or 3,
in the presence of at least one mol per mole of the amino diacid of an alkanesulphonic acid, optionally in the presence of a solvent.
The intermediate alkanesulphonates of the -benzyl esters of amino diacids and the -benzyl esters of amino diacids are obtained with a good yield and an excellent purity by virtue of this process. |
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