METHOD OF PREPARING EZETIMIBE AND INTERMEDIATE THEREOF

nd Disclosed is a method of preparing ezetimibe, including cross-metathesis using a Grubbs 2catalyst and deprotection using a Pearlman's catalyst, and an intermediate thereof. The method of preparing ezetimibe is useful as an efficient ezetimibe synthesis technique in pharmaceutical fields usin...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
1. Verfasser: Kangwon National University, University Industry Cooperation Foundation
Format: Patent
Sprache:eng
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:nd Disclosed is a method of preparing ezetimibe, including cross-metathesis using a Grubbs 2catalyst and deprotection using a Pearlman's catalyst, and an intermediate thereof. The method of preparing ezetimibe is useful as an efficient ezetimibe synthesis technique in pharmaceutical fields using ezetimibe as a raw material.