Copper-catalyzed borylative coupling of vinylazaarenes and -Boc imines
Cu-catalyzed three-component couplings of vinylazaarenes, B 2 (pin) 2 , and N -Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities. Diastereoselective Cu-catalyzed three-component...
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| Veröffentlicht in: | Chemical communications (Cambridge, England) England), 2016-02, Vol.52 (19), p.377-3772 |
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| Hauptverfasser: | , , |
| Format: | Artikel |
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| Online-Zugang: | Volltext |
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| Zusammenfassung: | Cu-catalyzed three-component couplings of vinylazaarenes, B
2
(pin)
2
, and
N
-Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities.
Diastereoselective Cu-catalyzed three-component couplings of vinylazaarenes, B
2
(pin)
2
, and
N
-Boc imines are described. |
|---|---|
| ISSN: | 1359-7345 1364-548X |
| DOI: | 10.1039/c6cc00603e |