Palladium-Catalyzed Regioselective C8–H Amination of 1‑Naphthylamine Derivatives with Aliphatic Amines

A simple and facile protocol for palladium-catalyzed picolinamide-directed C8–H amination of 1-naphthylamine derivatives with simple secondary aliphatic amines was developed, thereby providing a new route to 1,8-naphthalenediamine derivatives. It is noteworthy that the picolinamide moiety as a biden...

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Veröffentlicht in:	Organic letters 2016-09, Vol.18 (18), p.4594-4597
Hauptverfasser:	Li, Zexian, Sun, Suyan, Qiao, Huijie, Yang, Fan, Zhu, Yu, Kang, Jianxun, Wu, Yusheng, Wu, Yangjie
Format:	Artikel
Sprache:	eng
Schlagworte:	amination amines catalytic activity moieties palladium regioselectivity
Online-Zugang:	Volltext
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