Synthesis of amide libraries with immobilized HOBt
Highly reactive N-acylating solid-phase reagents based on macroporous polystyrene-bound 1-hydroxybenzotriazole (P-HOBt) and silica-bound 1-hydroxybenzotriazole (Si-HOBt) were prepared and compared for reactivity by synthesis of small combinatorial libraries of acetamides and benzamides.
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| Veröffentlicht in: | Tetrahedron letters 2011-05, Vol.52 (21), p.2722-2724 |
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| container_issue | 21 |
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| container_title | Tetrahedron letters |
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| creator | Vokkaliga, Smitha Jeong, Jeannie LaCourse, William R. Kalivretenos, Aristotle |
| description | Highly reactive N-acylating solid-phase reagents based on macroporous polystyrene-bound 1-hydroxybenzotriazole (P-HOBt) and silica-bound 1-hydroxybenzotriazole (Si-HOBt) were prepared and compared for reactivity by synthesis of small combinatorial libraries of acetamides and benzamides. |
| doi_str_mv | 10.1016/j.tetlet.2011.03.097 |
| format | Article |
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| ispartof | Tetrahedron letters, 2011-05, Vol.52 (21), p.2722-2724 |
| issn | 0040-4039 1873-3581 |
| language | eng |
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| source | Elsevier ScienceDirect Journals Complete |
| subjects | Aliphatic compounds Amide library Amides Benzamide Chemical reactivity Chemistry Combinatorial analysis Combinatorial library Exact sciences and technology Heterocyclic compounds Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings Libraries Organic chemistry Polymer-bound hydroxybenzotriazole Preparations and properties Reactivity and mechanisms Solid-phase synthesis Synthesis (chemistry) Tetrahedrons |
| title | Synthesis of amide libraries with immobilized HOBt |
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