Azetidine Iminosugars from the Cyclization of 3,5-Di-O-triflates of α-Furanosides and of 2,4-Di-O-triflates of β-Pyranosides Derived from Glucose

Azetidine Iminosugars from the Cyclization of 3,5-Di-O-triflates of α-Furanosides and of 2,4-Di-O-triflates of β-Pyranosides Derived from Glucose

Primary amines with either 3,5-di-O-ditriflates of α-furanosides or 2,4-di-O-triflates of β-pyranosides form bicyclic azetidines in high yield.

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Veröffentlicht in:Organic letters 2012-04, Vol.14 (8), p.2142-2145
Hauptverfasser: Lenagh-Snow, Gabriel M. J, Araújo, Noelia, Jenkinson, Sarah F, Martínez, R. Fernando, Shimada, Yousuke, Yu, Chu-Yi, Kato, Atsushi, Fleet, George W. J
Format: Artikel
Sprache:eng
Schlagworte:
Amines - chemistry
Azetidines - chemical synthesis
Azetidines - chemistry
Cyclization
Glucose - chemistry
Imino Sugars - chemical synthesis
Imino Sugars - chemistry
Mesylates - chemistry
Molecular Structure
Structure-Activity Relationship
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Beschreibung
Zusammenfassung:Primary amines with either 3,5-di-O-ditriflates of α-furanosides or 2,4-di-O-triflates of β-pyranosides form bicyclic azetidines in high yield.
ISSN:1523-7060
1523-7052
DOI:10.1021/ol300669v