Synthesis, photophysical, antibacterial and larvicidal studies on triazolophanes with 5-nitro isophthalate functionality at the intraannular position
1 : 1 and 2 : 2 oligomeric triazolophanes with 5-nitro isophthalate and triazolyl functionalities at the intraannular position have been synthesized by copper( i ) catalyzed 1,3 dipolar cycloaddition of the corresponding propargylic esters with various phenyl substituted aliphatic azides under mild...
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| Veröffentlicht in: | New journal of chemistry 2018, Vol.42 (15), p.12684-12691 |
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| container_issue | 15 |
| container_start_page | 12684 |
| container_title | New journal of chemistry |
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| creator | Selvarani, Sivasamy Rajakumar, Perumal Nagaraj, Subramani Choudhury, Manisha Velmurugan, Devadasan |
| description | 1 : 1 and 2 : 2 oligomeric triazolophanes with 5-nitro isophthalate and triazolyl functionalities at the intraannular position have been synthesized by copper(
i
) catalyzed 1,3 dipolar cycloaddition of the corresponding propargylic esters with various phenyl substituted aliphatic azides under mild conditions through click methodology. The 1 : 1 oligomeric triazolophanes exhibit good target binding ability and better antibacterial activity against
Staphylococcus aureus
,
Bacillus subtilis
,
Salmonella typhi
and
Escherichia coli
bacteria than the 2 : 2 oligomeric triazolophanes, supported by molecular docking studies, and triazolophanes T
3
, T
4
and T
5
show good larvicidal activity. |
| doi_str_mv | 10.1039/C8NJ01248B |
| format | Article |
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i
) catalyzed 1,3 dipolar cycloaddition of the corresponding propargylic esters with various phenyl substituted aliphatic azides under mild conditions through click methodology. The 1 : 1 oligomeric triazolophanes exhibit good target binding ability and better antibacterial activity against
Staphylococcus aureus
,
Bacillus subtilis
,
Salmonella typhi
and
Escherichia coli
bacteria than the 2 : 2 oligomeric triazolophanes, supported by molecular docking studies, and triazolophanes T
3
, T
4
and T
5
show good larvicidal activity.</description><identifier>ISSN: 1144-0546</identifier><identifier>EISSN: 1369-9261</identifier><identifier>DOI: 10.1039/C8NJ01248B</identifier><language>eng</language><publisher>Cambridge: Royal Society of Chemistry</publisher><subject>Aliphatic compounds ; Chemical synthesis ; Cycloaddition ; E coli ; Esters ; Molecular chains ; Molecular docking ; Salmonella</subject><ispartof>New journal of chemistry, 2018, Vol.42 (15), p.12684-12691</ispartof><rights>Copyright Royal Society of Chemistry 2018</rights><lds50>peer_reviewed</lds50><woscitedreferencessubscribed>false</woscitedreferencessubscribed><citedby>FETCH-LOGICAL-c259t-688120beaf8c49bdf8550c9dc0fa8e26722d940cb6325c0cc90df73f67aeaeb73</citedby><cites>FETCH-LOGICAL-c259t-688120beaf8c49bdf8550c9dc0fa8e26722d940cb6325c0cc90df73f67aeaeb73</cites><orcidid>0000-0001-5617-2942</orcidid></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><link.rule.ids>314,780,784,4024,27923,27924,27925</link.rule.ids></links><search><creatorcontrib>Selvarani, Sivasamy</creatorcontrib><creatorcontrib>Rajakumar, Perumal</creatorcontrib><creatorcontrib>Nagaraj, Subramani</creatorcontrib><creatorcontrib>Choudhury, Manisha</creatorcontrib><creatorcontrib>Velmurugan, Devadasan</creatorcontrib><title>Synthesis, photophysical, antibacterial and larvicidal studies on triazolophanes with 5-nitro isophthalate functionality at the intraannular position</title><title>New journal of chemistry</title><description>1 : 1 and 2 : 2 oligomeric triazolophanes with 5-nitro isophthalate and triazolyl functionalities at the intraannular position have been synthesized by copper(
i
) catalyzed 1,3 dipolar cycloaddition of the corresponding propargylic esters with various phenyl substituted aliphatic azides under mild conditions through click methodology. The 1 : 1 oligomeric triazolophanes exhibit good target binding ability and better antibacterial activity against
Staphylococcus aureus
,
Bacillus subtilis
,
Salmonella typhi
and
Escherichia coli
bacteria than the 2 : 2 oligomeric triazolophanes, supported by molecular docking studies, and triazolophanes T
3
, T
4
and T
5
show good larvicidal activity.</description><subject>Aliphatic compounds</subject><subject>Chemical synthesis</subject><subject>Cycloaddition</subject><subject>E coli</subject><subject>Esters</subject><subject>Molecular chains</subject><subject>Molecular docking</subject><subject>Salmonella</subject><issn>1144-0546</issn><issn>1369-9261</issn><fulltext>true</fulltext><rsrctype>article</rsrctype><creationdate>2018</creationdate><recordtype>article</recordtype><recordid>eNpFUMtOwzAQtBBIlMKFL7DEDTVgO4kTH6HiqQoOwDnaOLbiKtjBdkDlP_hfXBWJ0-7Mzs6uBqFTSi4oycXlsn56JJQV9fUemtGci0wwTvdTT4siI2XBD9FRCGtCKK04naGfl42NvQomLPDYu-jGfhOMhGGBwUbTgozKGxgS6vAA_tNI0yUY4tQZFbCzOKb5txvSJtjEfJnY4zKzJnqHTUh07GGAqLCerIzGWRhM3GCIOB3GxkYPYO2UzPHogtkqjtGBhiGok786R2-3N6_L-2z1fPewvFplkpUiZryuKSOtAl3LQrSdrsuSSNFJoqFWjFeMdaIgsuU5KyWRUpBOV7nmFShQbZXP0dnOd_TuY1IhNms3-fRgaBip8rIqBOdJdb5TSe9C8Eo3ozfv4DcNJc029uY_9vwXfxx6Cg</recordid><startdate>2018</startdate><enddate>2018</enddate><creator>Selvarani, Sivasamy</creator><creator>Rajakumar, Perumal</creator><creator>Nagaraj, Subramani</creator><creator>Choudhury, Manisha</creator><creator>Velmurugan, Devadasan</creator><general>Royal Society of Chemistry</general><scope>AAYXX</scope><scope>CITATION</scope><scope>7SR</scope><scope>8BQ</scope><scope>8FD</scope><scope>H9R</scope><scope>JG9</scope><scope>KA0</scope><orcidid>https://orcid.org/0000-0001-5617-2942</orcidid></search><sort><creationdate>2018</creationdate><title>Synthesis, photophysical, antibacterial and larvicidal studies on triazolophanes with 5-nitro isophthalate functionality at the intraannular position</title><author>Selvarani, Sivasamy ; Rajakumar, Perumal ; Nagaraj, Subramani ; Choudhury, Manisha ; Velmurugan, Devadasan</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-LOGICAL-c259t-688120beaf8c49bdf8550c9dc0fa8e26722d940cb6325c0cc90df73f67aeaeb73</frbrgroupid><rsrctype>articles</rsrctype><prefilter>articles</prefilter><language>eng</language><creationdate>2018</creationdate><topic>Aliphatic compounds</topic><topic>Chemical synthesis</topic><topic>Cycloaddition</topic><topic>E coli</topic><topic>Esters</topic><topic>Molecular chains</topic><topic>Molecular docking</topic><topic>Salmonella</topic><toplevel>peer_reviewed</toplevel><toplevel>online_resources</toplevel><creatorcontrib>Selvarani, Sivasamy</creatorcontrib><creatorcontrib>Rajakumar, Perumal</creatorcontrib><creatorcontrib>Nagaraj, Subramani</creatorcontrib><creatorcontrib>Choudhury, Manisha</creatorcontrib><creatorcontrib>Velmurugan, Devadasan</creatorcontrib><collection>CrossRef</collection><collection>Engineered Materials Abstracts</collection><collection>METADEX</collection><collection>Technology Research Database</collection><collection>Illustrata: Natural Sciences</collection><collection>Materials Research Database</collection><collection>ProQuest Illustrata: Technology Collection</collection><jtitle>New journal of chemistry</jtitle></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext</fulltext></delivery><addata><au>Selvarani, Sivasamy</au><au>Rajakumar, Perumal</au><au>Nagaraj, Subramani</au><au>Choudhury, Manisha</au><au>Velmurugan, Devadasan</au><format>journal</format><genre>article</genre><ristype>JOUR</ristype><atitle>Synthesis, photophysical, antibacterial and larvicidal studies on triazolophanes with 5-nitro isophthalate functionality at the intraannular position</atitle><jtitle>New journal of chemistry</jtitle><date>2018</date><risdate>2018</risdate><volume>42</volume><issue>15</issue><spage>12684</spage><epage>12691</epage><pages>12684-12691</pages><issn>1144-0546</issn><eissn>1369-9261</eissn><abstract>1 : 1 and 2 : 2 oligomeric triazolophanes with 5-nitro isophthalate and triazolyl functionalities at the intraannular position have been synthesized by copper(
i
) catalyzed 1,3 dipolar cycloaddition of the corresponding propargylic esters with various phenyl substituted aliphatic azides under mild conditions through click methodology. The 1 : 1 oligomeric triazolophanes exhibit good target binding ability and better antibacterial activity against
Staphylococcus aureus
,
Bacillus subtilis
,
Salmonella typhi
and
Escherichia coli
bacteria than the 2 : 2 oligomeric triazolophanes, supported by molecular docking studies, and triazolophanes T
3
, T
4
and T
5
show good larvicidal activity.</abstract><cop>Cambridge</cop><pub>Royal Society of Chemistry</pub><doi>10.1039/C8NJ01248B</doi><tpages>8</tpages><orcidid>https://orcid.org/0000-0001-5617-2942</orcidid></addata></record> |
| fulltext | fulltext |
| identifier | ISSN: 1144-0546 |
| ispartof | New journal of chemistry, 2018, Vol.42 (15), p.12684-12691 |
| issn | 1144-0546 1369-9261 |
| language | eng |
| recordid | cdi_proquest_journals_2073574966 |
| source | Royal Society Of Chemistry Journals 2008-; Alma/SFX Local Collection |
| subjects | Aliphatic compounds Chemical synthesis Cycloaddition E coli Esters Molecular chains Molecular docking Salmonella |
| title | Synthesis, photophysical, antibacterial and larvicidal studies on triazolophanes with 5-nitro isophthalate functionality at the intraannular position |
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