Synthesis, Antifungal Activity, and SAR Study of Some New 6‐Perfluoropropanyl Quinoline Derivatives

A series of novel quinoline derivatives containing perfluoropropanyl moiety were designed and synthesized. The bioassay results showed that some of them exhibited good control efficacy against Pyricularia oryae. The fungicidal activity was affected by the substituted position in the molecule. It was...

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Veröffentlicht in:Journal of heterocyclic chemistry 2018-01, Vol.55 (1), p.240-245
Hauptverfasser: Fang, Yue‐Ming, Zhang, Rui‐Rui, Shen, Zhong‐Hua, Wu, Hong‐Ke, Tan, Cheng‐Xia, Weng, Jian‐Quan, Xu, Tian‐Ming, Liu, Xing‐Hai
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Sprache:eng
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Zusammenfassung:A series of novel quinoline derivatives containing perfluoropropanyl moiety were designed and synthesized. The bioassay results showed that some of them exhibited good control efficacy against Pyricularia oryae. The fungicidal activity was affected by the substituted position in the molecule. It was found that the compound 3n possessed highest control effect against P. oryae at different concentration. It is better than that of control Tebufloquin.
ISSN:0022-152X
1943-5193
DOI:10.1002/jhet.3031