Microwave-assisted synthesis of bis(N-substituted thiazol-2-amine) derivatives and their biological activities
New 4,4′-(4,6-dimethoxy-1,3-phenylene)-bis( -substituted thiazol-2-amine) derivatives were synthesized from 1,1′-(4,6-dimethoxy-1,3-phenylene)-bis(2-bromoethanone) and substituted thioureas under conventional and microwave irradiation conditions. All products were subjected to antibacterial and anti...
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| Veröffentlicht in: | Heterocyclic communications 2017-10, Vol.23 (5), p.405-409 |
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| container_issue | 5 |
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| container_title | Heterocyclic communications |
| container_volume | 23 |
| creator | Baba, N.H. Kumar Ashok, D. Rao, Boddu Ananda Sarasija, Madderla Murthy, N.Y.S. Srinivasarao, Vankadari Parthasarathy, Tigulla |
| description | New 4,4′-(4,6-dimethoxy-1,3-phenylene)-bis(
-substituted thiazol-2-amine) derivatives
were synthesized from 1,1′-(4,6-dimethoxy-1,3-phenylene)-bis(2-bromoethanone)
and substituted thioureas
under conventional and microwave irradiation conditions. All products were subjected to
antibacterial and anti-TB evaluation. Some of the compounds exhibit good activities against
(+ve),
(−ve) strains and
H37Rv. |
| doi_str_mv | 10.1515/hc-2017-0129 |
| format | Article |
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-substituted thiazol-2-amine) derivatives
were synthesized from 1,1′-(4,6-dimethoxy-1,3-phenylene)-bis(2-bromoethanone)
and substituted thioureas
under conventional and microwave irradiation conditions. All products were subjected to
antibacterial and anti-TB evaluation. Some of the compounds exhibit good activities against
(+ve),
(−ve) strains and
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-substituted thiazol-2-amine) derivatives
were synthesized from 1,1′-(4,6-dimethoxy-1,3-phenylene)-bis(2-bromoethanone)
and substituted thioureas
under conventional and microwave irradiation conditions. All products were subjected to
antibacterial and anti-TB evaluation. Some of the compounds exhibit good activities against
(+ve),
(−ve) strains and
H37Rv.</description><subject>anti-TB</subject><subject>antibacterial</subject><subject>Derivatives</subject><subject>E coli</subject><subject>microwave irradiation</subject><subject>thiazole</subject><subject>Thioureas</subject><subject>Tuberculosis</subject><issn>0793-0283</issn><issn>2191-0197</issn><fulltext>true</fulltext><rsrctype>article</rsrctype><creationdate>2017</creationdate><recordtype>article</recordtype><recordid>eNptkE1LAzEQhoMoWGpv_oAFLwpGk-xmt_EmxS-oetFzyMdsm7LdrUm2pf56s9SDB-cyM8zzvgMvQueU3FBO-e3SYEZohQll4giNGBU0zaI6RiNSiRwTNs1P0SSEFUlVCMorMkLtqzO-26ktYBWCCxFsFvZtXEJasq7OtAuXbzj0OkQX--Ecl059dw1mWK1dC1eZBe-2KrothEy1AwDOJ2HXdAtnVJMpk44uOghn6KRWTYDJbx-jz8eHj9kznr8_vczu59jknEVMSW0tq5TShS5ppW3ONBWmVHXBamErO-WclQAWjKk00IKURhtqp8zaohQ2H6OLg-_Gd189hChXXe_b9FJSwUkSc1Em6vpApQhC8FDLjXdr5feSEjmEKpdGDqHKIdSE3x3wnWoieAsL3-_T8Mf7HxnLeUF4_gND-H9W</recordid><startdate>20171026</startdate><enddate>20171026</enddate><creator>Baba, N.H. Kumar</creator><creator>Ashok, D.</creator><creator>Rao, Boddu Ananda</creator><creator>Sarasija, Madderla</creator><creator>Murthy, N.Y.S.</creator><creator>Srinivasarao, Vankadari</creator><creator>Parthasarathy, Tigulla</creator><general>De Gruyter</general><general>Walter de Gruyter GmbH</general><scope>AAYXX</scope><scope>CITATION</scope></search><sort><creationdate>20171026</creationdate><title>Microwave-assisted synthesis of bis(N-substituted thiazol-2-amine) derivatives and their biological activities</title><author>Baba, N.H. Kumar ; Ashok, D. ; Rao, Boddu Ananda ; Sarasija, Madderla ; Murthy, N.Y.S. ; Srinivasarao, Vankadari ; Parthasarathy, Tigulla</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-LOGICAL-c352t-10fdd27aab4b617bd32b19c6af42f9d7d85526eedecc7be1406cbc1d82dd469d3</frbrgroupid><rsrctype>articles</rsrctype><prefilter>articles</prefilter><language>eng</language><creationdate>2017</creationdate><topic>anti-TB</topic><topic>antibacterial</topic><topic>Derivatives</topic><topic>E coli</topic><topic>microwave irradiation</topic><topic>thiazole</topic><topic>Thioureas</topic><topic>Tuberculosis</topic><toplevel>peer_reviewed</toplevel><toplevel>online_resources</toplevel><creatorcontrib>Baba, N.H. Kumar</creatorcontrib><creatorcontrib>Ashok, D.</creatorcontrib><creatorcontrib>Rao, Boddu Ananda</creatorcontrib><creatorcontrib>Sarasija, Madderla</creatorcontrib><creatorcontrib>Murthy, N.Y.S.</creatorcontrib><creatorcontrib>Srinivasarao, Vankadari</creatorcontrib><creatorcontrib>Parthasarathy, Tigulla</creatorcontrib><collection>CrossRef</collection><jtitle>Heterocyclic communications</jtitle></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext</fulltext></delivery><addata><au>Baba, N.H. Kumar</au><au>Ashok, D.</au><au>Rao, Boddu Ananda</au><au>Sarasija, Madderla</au><au>Murthy, N.Y.S.</au><au>Srinivasarao, Vankadari</au><au>Parthasarathy, Tigulla</au><format>journal</format><genre>article</genre><ristype>JOUR</ristype><atitle>Microwave-assisted synthesis of bis(N-substituted thiazol-2-amine) derivatives and their biological activities</atitle><jtitle>Heterocyclic communications</jtitle><date>2017-10-26</date><risdate>2017</risdate><volume>23</volume><issue>5</issue><spage>405</spage><epage>409</epage><pages>405-409</pages><issn>0793-0283</issn><eissn>2191-0197</eissn><abstract>New 4,4′-(4,6-dimethoxy-1,3-phenylene)-bis(
-substituted thiazol-2-amine) derivatives
were synthesized from 1,1′-(4,6-dimethoxy-1,3-phenylene)-bis(2-bromoethanone)
and substituted thioureas
under conventional and microwave irradiation conditions. All products were subjected to
antibacterial and anti-TB evaluation. Some of the compounds exhibit good activities against
(+ve),
(−ve) strains and
H37Rv.</abstract><cop>Berlin</cop><pub>De Gruyter</pub><doi>10.1515/hc-2017-0129</doi><tpages>5</tpages><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext |
| identifier | ISSN: 0793-0283 |
| ispartof | Heterocyclic communications, 2017-10, Vol.23 (5), p.405-409 |
| issn | 0793-0283 2191-0197 |
| language | eng |
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| source | Elektronische Zeitschriftenbibliothek - Frei zugängliche E-Journals; Walter De Gruyter: Open Access Journals |
| subjects | anti-TB antibacterial Derivatives E coli microwave irradiation thiazole Thioureas Tuberculosis |
| title | Microwave-assisted synthesis of bis(N-substituted thiazol-2-amine) derivatives and their biological activities |
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