ChemInform Abstract: Synthesis of Indole‐Annulated Sulfur Heterocycles Using Copper‐Catalyzed C—N Coupling and Palladium‐Catalyzed Direct Arylation

Biologically relevant benzothiazinoindoles and isothiochromenoindoles are prepared using Cu‐catalyzed Ullmann‐type coupling and Pd‐catalyzed arylation, respectively, as key steps to construct the polycyclic frameworks.

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Bibliographische Detailangaben
Veröffentlicht in:	ChemInform 2016-07, Vol.47 (31), p.no-no
Hauptverfasser:	Shelke, Ganesh M., Jha, Mukund, Kumar, Anil
Format:	Artikel
Sprache:	eng
Schlagworte:	amination, N‐alkylation, N‐arylation catalysis, phase‐transfer catalysis fused pyrrole derivatives ring closure reactions, annulation reactions sulfuration, sulfonation, S‐alkylation thiazine derivatives
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Beschreibung
Zusammenfassung:	Biologically relevant benzothiazinoindoles and isothiochromenoindoles are prepared using Cu‐catalyzed Ullmann‐type coupling and Pd‐catalyzed arylation, respectively, as key steps to construct the polycyclic frameworks.
ISSN:	0931-7597 1522-2667
DOI:	10.1002/chin.201631154