Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one

Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one

Synthesis of new 1,2-dihydro-3 H -pyrazolo[3,4- d ] pyrimidin-3-ones 4–6 starting with ethyl 4-hydroxy-2-methylthio-pyrimidine-5-carboxylate ( 1 ) under classical heating and microwave-induced conditions is reported. The antibacterial activities of the synthesized compounds were evaluated using chlo...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Veröffentlicht in:Heterocyclic communications 2016-02, Vol.22 (1), p.49-53
Hauptverfasser: Ebrahimpour, Zahra, Shiri, Ali, Bakavoli, Mehdi, Seyedi, Seyed Mohammad, Bahreini, Masoumeh, Oroojalian, Fatemeh
Format: Artikel
Sprache:eng
Schlagworte:
Chemical synthesis
Microwaves
Pharmacology
Online-Zugang:Volltext
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
container_end_page 53
container_issue 1
container_start_page 49
container_title Heterocyclic communications
container_volume 22
creator Ebrahimpour, Zahra
Shiri, Ali
Bakavoli, Mehdi
Seyedi, Seyed Mohammad
Bahreini, Masoumeh
Oroojalian, Fatemeh
description Synthesis of new 1,2-dihydro-3 H -pyrazolo[3,4- d ] pyrimidin-3-ones 4–6 starting with ethyl 4-hydroxy-2-methylthio-pyrimidine-5-carboxylate ( 1 ) under classical heating and microwave-induced conditions is reported. The antibacterial activities of the synthesized compounds were evaluated using chloramphenicol and streptomycin as reference drugs.
doi_str_mv 10.1515/hc-2015-0145
format Article
fullrecord <record><control><sourceid>proquest_cross</sourceid><recordid>TN_cdi_proquest_journals_1762942998</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>3945439381</sourcerecordid><originalsourceid>FETCH-LOGICAL-c658-f79d9e5195dd32f3252c378beb4571180edd2ed8ad1ec0a07fc7c47985f229f33</originalsourceid><addsrcrecordid>eNotkE1LAzEQhoMoWGpv_oCA10bzsWk2RylqhYqX3kRCmg82Zd3UZLtlvfnPTakDw8y8M8wMDwC3BN8TTvhDYxDFhCNMKn4BJpRIUnIpLsEEC8kQpjW7BrOcd7hYJQkXeAJ-34JJ8agHh3TOIffOwjx2feNKAXVni_dhq03vUtAtdINuD7oPsYPRw84doS2NoSiDyyeJzCmyoRltiojBFUT7Memf2MYPNq8QtPCzCOEr2NAhhmLnbsCV1212s_84BZvnp81yhdbvL6_LxzUyC14jL6SVjhPJrWXUM8qpYaLeum3FBSE1dtZSZ2ttiTNYY-GNMJWQNfeUSs_YFNyd1-5T_D643KtdPKSuXFRELKisqJR1mZqfpwqUnJPzal-e1WlUBKsTZtUYdcKsTpjZH9a8cAU</addsrcrecordid><sourcetype>Aggregation Database</sourcetype><iscdi>true</iscdi><recordtype>article</recordtype><pqid>1762942998</pqid></control><display><type>article</type><title>Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one</title><source>De Gruyter Open Access Journals</source><source>Elektronische Zeitschriftenbibliothek - Frei zugängliche E-Journals</source><creator>Ebrahimpour, Zahra ; Shiri, Ali ; Bakavoli, Mehdi ; Seyedi, Seyed Mohammad ; Bahreini, Masoumeh ; Oroojalian, Fatemeh</creator><creatorcontrib>Ebrahimpour, Zahra ; Shiri, Ali ; Bakavoli, Mehdi ; Seyedi, Seyed Mohammad ; Bahreini, Masoumeh ; Oroojalian, Fatemeh</creatorcontrib><description>Synthesis of new 1,2-dihydro-3 H -pyrazolo[3,4- d ] pyrimidin-3-ones 4–6 starting with ethyl 4-hydroxy-2-methylthio-pyrimidine-5-carboxylate ( 1 ) under classical heating and microwave-induced conditions is reported. The antibacterial activities of the synthesized compounds were evaluated using chloramphenicol and streptomycin as reference drugs.</description><identifier>ISSN: 0793-0283</identifier><identifier>EISSN: 2191-0197</identifier><identifier>DOI: 10.1515/hc-2015-0145</identifier><language>eng</language><publisher>Berlin: Walter de Gruyter GmbH</publisher><subject>Chemical synthesis ; Microwaves ; Pharmacology</subject><ispartof>Heterocyclic communications, 2016-02, Vol.22 (1), p.49-53</ispartof><rights>Copyright Walter de Gruyter GmbH Feb 2016</rights><lds50>peer_reviewed</lds50><woscitedreferencessubscribed>false</woscitedreferencessubscribed><cites>FETCH-LOGICAL-c658-f79d9e5195dd32f3252c378beb4571180edd2ed8ad1ec0a07fc7c47985f229f33</cites></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><link.rule.ids>314,776,780,27901,27902</link.rule.ids></links><search><creatorcontrib>Ebrahimpour, Zahra</creatorcontrib><creatorcontrib>Shiri, Ali</creatorcontrib><creatorcontrib>Bakavoli, Mehdi</creatorcontrib><creatorcontrib>Seyedi, Seyed Mohammad</creatorcontrib><creatorcontrib>Bahreini, Masoumeh</creatorcontrib><creatorcontrib>Oroojalian, Fatemeh</creatorcontrib><title>Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one</title><title>Heterocyclic communications</title><description>Synthesis of new 1,2-dihydro-3 H -pyrazolo[3,4- d ] pyrimidin-3-ones 4–6 starting with ethyl 4-hydroxy-2-methylthio-pyrimidine-5-carboxylate ( 1 ) under classical heating and microwave-induced conditions is reported. The antibacterial activities of the synthesized compounds were evaluated using chloramphenicol and streptomycin as reference drugs.</description><subject>Chemical synthesis</subject><subject>Microwaves</subject><subject>Pharmacology</subject><issn>0793-0283</issn><issn>2191-0197</issn><fulltext>true</fulltext><rsrctype>article</rsrctype><creationdate>2016</creationdate><recordtype>article</recordtype><recordid>eNotkE1LAzEQhoMoWGpv_oCA10bzsWk2RylqhYqX3kRCmg82Zd3UZLtlvfnPTakDw8y8M8wMDwC3BN8TTvhDYxDFhCNMKn4BJpRIUnIpLsEEC8kQpjW7BrOcd7hYJQkXeAJ-34JJ8agHh3TOIffOwjx2feNKAXVni_dhq03vUtAtdINuD7oPsYPRw84doS2NoSiDyyeJzCmyoRltiojBFUT7Memf2MYPNq8QtPCzCOEr2NAhhmLnbsCV1212s_84BZvnp81yhdbvL6_LxzUyC14jL6SVjhPJrWXUM8qpYaLeum3FBSE1dtZSZ2ttiTNYY-GNMJWQNfeUSs_YFNyd1-5T_D643KtdPKSuXFRELKisqJR1mZqfpwqUnJPzal-e1WlUBKsTZtUYdcKsTpjZH9a8cAU</recordid><startdate>20160201</startdate><enddate>20160201</enddate><creator>Ebrahimpour, Zahra</creator><creator>Shiri, Ali</creator><creator>Bakavoli, Mehdi</creator><creator>Seyedi, Seyed Mohammad</creator><creator>Bahreini, Masoumeh</creator><creator>Oroojalian, Fatemeh</creator><general>Walter de Gruyter GmbH</general><scope>AAYXX</scope><scope>CITATION</scope></search><sort><creationdate>20160201</creationdate><title>Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one</title><author>Ebrahimpour, Zahra ; Shiri, Ali ; Bakavoli, Mehdi ; Seyedi, Seyed Mohammad ; Bahreini, Masoumeh ; Oroojalian, Fatemeh</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-LOGICAL-c658-f79d9e5195dd32f3252c378beb4571180edd2ed8ad1ec0a07fc7c47985f229f33</frbrgroupid><rsrctype>articles</rsrctype><prefilter>articles</prefilter><language>eng</language><creationdate>2016</creationdate><topic>Chemical synthesis</topic><topic>Microwaves</topic><topic>Pharmacology</topic><toplevel>peer_reviewed</toplevel><toplevel>online_resources</toplevel><creatorcontrib>Ebrahimpour, Zahra</creatorcontrib><creatorcontrib>Shiri, Ali</creatorcontrib><creatorcontrib>Bakavoli, Mehdi</creatorcontrib><creatorcontrib>Seyedi, Seyed Mohammad</creatorcontrib><creatorcontrib>Bahreini, Masoumeh</creatorcontrib><creatorcontrib>Oroojalian, Fatemeh</creatorcontrib><collection>CrossRef</collection><jtitle>Heterocyclic communications</jtitle></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext</fulltext></delivery><addata><au>Ebrahimpour, Zahra</au><au>Shiri, Ali</au><au>Bakavoli, Mehdi</au><au>Seyedi, Seyed Mohammad</au><au>Bahreini, Masoumeh</au><au>Oroojalian, Fatemeh</au><format>journal</format><genre>article</genre><ristype>JOUR</ristype><atitle>Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one</atitle><jtitle>Heterocyclic communications</jtitle><date>2016-02-01</date><risdate>2016</risdate><volume>22</volume><issue>1</issue><spage>49</spage><epage>53</epage><pages>49-53</pages><issn>0793-0283</issn><eissn>2191-0197</eissn><abstract>Synthesis of new 1,2-dihydro-3 H -pyrazolo[3,4- d ] pyrimidin-3-ones 4–6 starting with ethyl 4-hydroxy-2-methylthio-pyrimidine-5-carboxylate ( 1 ) under classical heating and microwave-induced conditions is reported. The antibacterial activities of the synthesized compounds were evaluated using chloramphenicol and streptomycin as reference drugs.</abstract><cop>Berlin</cop><pub>Walter de Gruyter GmbH</pub><doi>10.1515/hc-2015-0145</doi><tpages>5</tpages></addata></record>
fulltext fulltext
identifier ISSN: 0793-0283
ispartof Heterocyclic communications, 2016-02, Vol.22 (1), p.49-53
issn 0793-0283
2191-0197
language eng
recordid cdi_proquest_journals_1762942998
source De Gruyter Open Access Journals; Elektronische Zeitschriftenbibliothek - Frei zugängliche E-Journals
subjects Chemical synthesis
Microwaves
Pharmacology
title Microwave-assisted synthesis and antibacterial evaluation of new derivatives of 1,2-dihydro-3 H -pyrazolo[3,4- d ]pyrimidin-3-one
url https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-03T08%3A52%3A17IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-proquest_cross&rft_val_fmt=info:ofi/fmt:kev:mtx:journal&rft.genre=article&rft.atitle=Microwave-assisted%20synthesis%20and%20antibacterial%20evaluation%20of%20new%20derivatives%20of%201,2-dihydro-3%20H%20-pyrazolo%5B3,4-%20d%20%5Dpyrimidin-3-one&rft.jtitle=Heterocyclic%20communications&rft.au=Ebrahimpour,%20Zahra&rft.date=2016-02-01&rft.volume=22&rft.issue=1&rft.spage=49&rft.epage=53&rft.pages=49-53&rft.issn=0793-0283&rft.eissn=2191-0197&rft_id=info:doi/10.1515/hc-2015-0145&rft_dat=%3Cproquest_cross%3E3945439381%3C/proquest_cross%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_pqid=1762942998&rft_id=info:pmid/&rfr_iscdi=true