Cross-Coupling Reactions of Pyrimidin-2-yl Sulfonates with Phenols and Anilines： An Efficient Approach to C2-Functionalized Pyrimidines

Pyrimidin-2-yl sulfonates, as an efficient reaction partner, which can be easily prepared from cheap commercial materials, were coupled with phenols and anilines to give a wide array of C2-aryloxy- and arylaminopyrimidines in good to excellent yields under mild reaction conditions.

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Bibliographische Detailangaben
Veröffentlicht in:	Chinese journal of chemistry 2013-12, Vol.31 (12), p.1495-1502
Hauptverfasser:	Quan, Zhengjun, Jing, Fuqiang, Zhang, Zhang, Da, Yuxia, Wang, Xicun
Format:	Artikel
Sprache:	eng
Schlagworte:	C2-arylaminopyrimidines C2-aryloxypyrimidines cross-coupling Phenols pyrimindine-2-yl sulfonates 交叉偶联反应化合物反应条件嘧啶磺酰基磺酸盐苯胺类苯酚
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Beschreibung
Zusammenfassung:	Pyrimidin-2-yl sulfonates, as an efficient reaction partner, which can be easily prepared from cheap commercial materials, were coupled with phenols and anilines to give a wide array of C2-aryloxy- and arylaminopyrimidines in good to excellent yields under mild reaction conditions.
ISSN:	1001-604X 1614-7065
DOI:	10.1002/cjoc.201300536