Synthesis of 1-Triazolyl-4-trimethylsilyl-2-butanol and 1-Triazolyl-5-trimethylsilyl-2-pentanol Derivatives and an Investigation of Their Fungicidal Activities

A new series of azole derivatives of 1-triazolyl-4-trimethylsilyl-2-butanol and 1-triazolyl-5-trimethylsilyl-2-pentanol were synthesized and evaluated for fungicidal activities against rice blast, sheath blight, and powdery mildew on barley. The derivatives of 2,4-difluorobenzene exhibited high anti...

Ausführliche Beschreibung

Gespeichert in:

Bibliographische Detailangaben
Veröffentlicht in:	Chemical & pharmaceutical bulletin 2003, Vol.51(9), pp.1113-1116
Hauptverfasser:	Itoh, Hiroyuki, Yoneda, Rieko, Tobitsuka, Junzo, Ohta, Hiroshi, Takahi, Yukiyoshi, Tsuda, Mikio, Takeshiba, Hideo
Format:	Artikel
Sprache:	eng
Schlagworte:	1H-1,2,4-triazole Ascomycota - drug effects Biological and medical sciences Chemical control Control Fundamental and applied biological sciences. Psychology Fungal plant pathogens fungicidal activity Fungicides, Industrial - chemical synthesis Fungicides, Industrial - pharmacology Hordeum Magnetic Resonance Spectroscopy Oryza - microbiology Phytopathology. Animal pests. Plant and forest protection Plant Diseases - microbiology Rhizoctonia - drug effects silicon Spectrophotometry, Infrared synthesis Triazoles - chemical synthesis Triazoles - pharmacology Trimethylsilyl Compounds - chemical synthesis Trimethylsilyl Compounds - pharmacology
Online-Zugang:	Volltext
Tags:	Tag hinzufügen Keine Tags, Fügen Sie den ersten Tag hinzu!

Beschreibung
Zusammenfassung:	A new series of azole derivatives of 1-triazolyl-4-trimethylsilyl-2-butanol and 1-triazolyl-5-trimethylsilyl-2-pentanol were synthesized and evaluated for fungicidal activities against rice blast, sheath blight, and powdery mildew on barley. The derivatives of 2,4-difluorobenzene exhibited high antifungal activities when applied by spray, but exhibited no fungicidal activity by submerged application.
ISSN:	0009-2363 1347-5223
DOI:	10.1248/cpb.51.1113