A Novel Synthesis of 4-Aryl-and 4-Heteroarylpyridines via Diethyl (4-pyridyl) borane

A convenient method for the preparation of 4-aryl- and 4-heteroarylpyridines by the palladium-catalyzed cross-coupling reaction of diethyl (4-pyridyl) borane with aryl and heteroaryl halides is described.

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Bibliographische Detailangaben
Veröffentlicht in:	Chemical & pharmaceutical bulletin 1985/11/25, Vol.33(11), pp.4755-4763
Hauptverfasser:	ISHIKURA, MINORU, OHTA, TSUKASA, TERASHIMA, MASANAO
Format:	Artikel
Sprache:	eng
Schlagworte:	Chemistry Exact sciences and technology Heterocyclic compounds Heterocyclic compounds with only one n hetero atom and condensed derivatives Organic chemistry palladium-catalyzed cross-coupling reaction Preparations and properties
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Beschreibung
Zusammenfassung:	A convenient method for the preparation of 4-aryl- and 4-heteroarylpyridines by the palladium-catalyzed cross-coupling reaction of diethyl (4-pyridyl) borane with aryl and heteroaryl halides is described.
ISSN:	0009-2363 1347-5223
DOI:	10.1248/cpb.33.4755