Convenient access to C-2 or C-5 substituted 4-azaindole derivatives

Convenient access to C-2 or C-5 substituted 4-azaindole derivatives

Functionalization at C-2 and C-5 of N-benzenesulfonyl-4-azaindole 1 was performed by lithiation reactions and original palladium-catalyzed chemistry. It led to very useful new substituted 4-azaindole derivatives in fair to high yields. [Display omitted]

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Bibliographische Detailangaben
Veröffentlicht in:Tetrahedron 2010, Vol.66 (1), p.102-110
Hauptverfasser: Saab, Fabienne, Bénéteau, Valérie, Schoentgen, Françoise, Mérour, Jean-Yves, Routier, Sylvain
Format: Artikel
Sprache:eng
Schlagworte:
Biochemistry, Molecular Biology
Chemistry
Exact sciences and technology
Heterocyclic compounds
Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings
Life Sciences
Organic chemistry
Preparations and properties
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Beschreibung
Zusammenfassung:Functionalization at C-2 and C-5 of N-benzenesulfonyl-4-azaindole 1 was performed by lithiation reactions and original palladium-catalyzed chemistry. It led to very useful new substituted 4-azaindole derivatives in fair to high yields. [Display omitted]
ISSN:0040-4020
1464-5416
DOI:10.1016/j.tet.2009.11.040