A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF
The present disclosure provides a process of preparation of an antibacterial compound of Formula I, (S)-6-(5-(((2-(7-fluoro-l- methyl-2-oxo-l,2-dihydroquinolin-8-yl) ethyl) amino) methyl)-2- oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one formate salt. The present disclosure also provi...
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| creator | PEER MOHAMED, Shahul Hameed TUMMA, Harikrishna KAUSHIK KOTAKONDA, Harish |
| description | The present disclosure provides a process of preparation of an antibacterial compound of Formula I, (S)-6-(5-(((2-(7-fluoro-l- methyl-2-oxo-l,2-dihydroquinolin-8-yl) ethyl) amino) methyl)-2- oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one formate salt. The present disclosure also provides intermediates of the compound of Formula I and their preparation. The present disclosure further provides a process of preparation of compound of Formula I with improved yield and high purity.
La présente divulgation propose un procédé de préparation d'un composé antibactérien de formule I, sel formiate (S)-6-(5-(((2-(7-fluoro-1-méthyl-2-oxo-1,2-dihydroquinoléin-8-yl) éthyl) amino) méthyl)-2-oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one. La présente divulgation propose également des intermédiaires du composé de formule I et leur préparation. La présente divulgation propose en outre un procédé de préparation d'un composé de formule I avec un rendement amélioré et une pureté élevée. |
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La présente divulgation propose un procédé de préparation d'un composé antibactérien de formule I, sel formiate (S)-6-(5-(((2-(7-fluoro-1-méthyl-2-oxo-1,2-dihydroquinoléin-8-yl) éthyl) amino) méthyl)-2-oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one. La présente divulgation propose également des intermédiaires du composé de formule I et leur préparation. La présente divulgation propose en outre un procédé de préparation d'un composé de formule I avec un rendement amélioré et une pureté élevée.</description><language>eng ; fre</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; METALLURGY ; ORGANIC CHEMISTRY</subject><creationdate>2024</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20241212&DB=EPODOC&CC=WO&NR=2024252423A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20241212&DB=EPODOC&CC=WO&NR=2024252423A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>PEER MOHAMED, Shahul Hameed</creatorcontrib><creatorcontrib>TUMMA, Harikrishna</creatorcontrib><creatorcontrib>KAUSHIK KOTAKONDA, Harish</creatorcontrib><title>A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF</title><description>The present disclosure provides a process of preparation of an antibacterial compound of Formula I, (S)-6-(5-(((2-(7-fluoro-l- methyl-2-oxo-l,2-dihydroquinolin-8-yl) ethyl) amino) methyl)-2- oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one formate salt. The present disclosure also provides intermediates of the compound of Formula I and their preparation. The present disclosure further provides a process of preparation of compound of Formula I with improved yield and high purity.
La présente divulgation propose un procédé de préparation d'un composé antibactérien de formule I, sel formiate (S)-6-(5-(((2-(7-fluoro-1-méthyl-2-oxo-1,2-dihydroquinoléin-8-yl) éthyl) amino) méthyl)-2-oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one. La présente divulgation propose également des intermédiaires du composé de formule I et leur préparation. La présente divulgation propose en outre un procédé de préparation d'un composé de formule I avec un rendement amélioré et une pureté élevée.</description><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2024</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNSksKwjAQzcaFqHcYcC1oqgcYkwkN2ExIprgsReJKtFDvjxE8gPAe77tUGSEmNpQzsKuWIiYUz-EbMVSIP6MRSh4vYLiL3AdbawteMvhQl46sR6EM0lIidmu1uI-PuWx-ulJbR2LaXZleQ5mn8Vae5T1cWe_1UZ8qGzw0_70-nocwkg</recordid><startdate>20241212</startdate><enddate>20241212</enddate><creator>PEER MOHAMED, Shahul Hameed</creator><creator>TUMMA, Harikrishna</creator><creator>KAUSHIK KOTAKONDA, Harish</creator><scope>EVB</scope></search><sort><creationdate>20241212</creationdate><title>A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF</title><author>PEER MOHAMED, Shahul Hameed ; TUMMA, Harikrishna ; KAUSHIK KOTAKONDA, Harish</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2024252423A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2024</creationdate><topic>ACYCLIC OR CARBOCYCLIC COMPOUNDS</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><toplevel>online_resources</toplevel><creatorcontrib>PEER MOHAMED, Shahul Hameed</creatorcontrib><creatorcontrib>TUMMA, Harikrishna</creatorcontrib><creatorcontrib>KAUSHIK KOTAKONDA, Harish</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>PEER MOHAMED, Shahul Hameed</au><au>TUMMA, Harikrishna</au><au>KAUSHIK KOTAKONDA, Harish</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF</title><date>2024-12-12</date><risdate>2024</risdate><abstract>The present disclosure provides a process of preparation of an antibacterial compound of Formula I, (S)-6-(5-(((2-(7-fluoro-l- methyl-2-oxo-l,2-dihydroquinolin-8-yl) ethyl) amino) methyl)-2- oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one formate salt. The present disclosure also provides intermediates of the compound of Formula I and their preparation. The present disclosure further provides a process of preparation of compound of Formula I with improved yield and high purity.
La présente divulgation propose un procédé de préparation d'un composé antibactérien de formule I, sel formiate (S)-6-(5-(((2-(7-fluoro-1-méthyl-2-oxo-1,2-dihydroquinoléin-8-yl) éthyl) amino) méthyl)-2-oxooxazolidin-3-yl)-2H-pyrazino[2,3-b] [1,4] oxazin-3(4H)-one. La présente divulgation propose également des intermédiaires du composé de formule I et leur préparation. La présente divulgation propose en outre un procédé de préparation d'un composé de formule I avec un rendement amélioré et une pureté élevée.</abstract><oa>free_for_read</oa></addata></record> |
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| title | A PROCESS OF PREPARATION OF AN ANTIBACTERIAL COMPOUND AND ITS INTERMEDIATES THEREOF |
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