FORMULATIONS OF 19-NOR C3,3- DISUBSTITUTED C21-N-PYRAZOLYL STEROID AND METHODS OF USE THEREOF

This invention relates to a 19-nor C3,3-disubstituted C21-pyrazolyl steroid of formula (I) and pharmaceutical compositions thereof. Also disclosed herein are methods of making the pharmaceutical compositions of the 19-nor C3,3-disubstituted C21-pyrazolyl steroid of formula (I) and methods of using t...

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Bibliographische Detailangaben
Hauptverfasser:	NARAYAN, Padma, WILKERSON, Carolyn, WATSON, Paul, MENG, Jianing, CHEN, Xiaoxia, STUTZMAN, Todd, BERNER, Bret, JAIN, Raj
Format:	Patent
Sprache:	eng ; fre
Schlagworte:	HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:	This invention relates to a 19-nor C3,3-disubstituted C21-pyrazolyl steroid of formula (I) and pharmaceutical compositions thereof. Also disclosed herein are methods of making the pharmaceutical compositions of the 19-nor C3,3-disubstituted C21-pyrazolyl steroid of formula (I) and methods of using the 19-nor C3,3-disubstituted C21-pyrazolyl steroid of formula (I) or crystalline solid forms, pharmaceutically acceptable salts, and pharmaceutically acceptable compositions thereof. La présente invention concerne un stéroïde C21-pyrazolyle 19-nor C3,3-disubstitué de formule (I) et ses compositions pharmaceutiques. L'invention porte également sur des procédés de fabrication de compositions pharmaceutiques du stéroïde C21-pyrazolyle 19-nor C3,3-disubstitué de formule (I) et sur des procédés d'utilisation du stéroïde C21-pyrazolyle 19-nor C3,3-disubstitué de formule (I) ou de formes solides cristallines, des sels pharmaceutiquement acceptables et de leurs compositions pharmaceutiquement acceptables.