BICYCLIC HETEROCYCLES AS FGFR INHIBITORS

The present disclosure relates to bicyclic heterocycles, and pharmaceutical compositions of the same, that are inhibitors of the FGFR enzyme and are useful in the treatment of FGFR-associated diseases such as cancer. La présente invention concerne des hétérocycles bicycliques, et des compositions ph...

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Hauptverfasser: ROACH, Jeremy, SHVARTSBART, Artem, YAO, Wenqing, WITTEN, Michael
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creator ROACH, Jeremy
SHVARTSBART, Artem
YAO, Wenqing
WITTEN, Michael
description The present disclosure relates to bicyclic heterocycles, and pharmaceutical compositions of the same, that are inhibitors of the FGFR enzyme and are useful in the treatment of FGFR-associated diseases such as cancer. La présente invention concerne des hétérocycles bicycliques, et des compositions pharmaceutiques les contenant, qui sont des inhibiteurs de l'enzyme FGFR et sont utiles dans le traitement de maladies associées au FGFR telles que le cancer.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title BICYCLIC HETEROCYCLES AS FGFR INHIBITORS
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