BENZAZEPINE DERIVATIVE ALCOHOLATE OR CRYSTAL THEREOF

BENZAZEPINE DERIVATIVE ALCOHOLATE OR CRYSTAL THEREOF

This invention provides an alcoholate of (S)-N-[(S)-1-hydroxypropan-2-yl]-4-methyl-1-[2-methyl-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1H-benzo[b]azepine-4-carboxamide represented by formula (I), or a crystal thereof, which is applicable as an active ingredient of a pharmaceutical dr...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: NAGAI Kazushige, SAITOH Yukiharu, KASUGAI Nobuyoshi
Format: Patent
Sprache:eng ; fre ; jpn
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:This invention provides an alcoholate of (S)-N-[(S)-1-hydroxypropan-2-yl]-4-methyl-1-[2-methyl-4-(3-methyl-1H-pyrazol-1-yl)benzoyl]-2,3,4,5-tetrahydro-1H-benzo[b]azepine-4-carboxamide represented by formula (I), or a crystal thereof, which is applicable as an active ingredient of a pharmaceutical drug. La présente invention concerne un alcoolate de (S)-N-[(S)-1-hydroxypropan-2-yl]-4-méthyl-1-[2-méthyl-4-(3-méthyl-1H-pyrazol-1-yl) benzoyl]-2,3,4,5-tétrahydro-1H-benzo[b]azépine-4-carboxamide représenté par la formule (I), ou un cristal de celui-ci, qui est utilisable en tant que principe actif d'un médicament pharmaceutique. 本発明は、医薬品の原薬としての利用可能性を有する、式（Ｉ）によって表される（Ｓ）－Ｎ－［（Ｓ）－１－ヒドロキシプロパン－２－イル］－４－メチル－１－［２－メチル－４－（３－メチル－１Ｈ－ピラゾール－１－イル）ベンゾイル］－２，３，４，５－テトラヒドロ－１Ｈ－ベンゾ［ｂ］アゼピン－４－カルボキサミドのアルコール和物又はその結晶を提供する。