NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS
The invention relates to novel heteroaryl and heterocycle compounds of formula I and pharmaceutical compositions comprising them, uses and methods thereof for inhibiting the activity of PI3K and for treating inflammatory and autoimmune diseases and cancer. La présente invention concerne de nouveaux...
Gespeichert in:
| Hauptverfasser: | , , , , , , , , , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | eng ; fre |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | LEBSACK, ALEC DONALD ECCLES, WENDY DAI, GUANGXIU CHAI, WENYING MEDUNA, STEVEN PAUL KEITH, JOHN MATTHEW VENABLE, JENNIFER DIANE WENG, JIANYANG SMITH, RUSSELL CHRISTOPHER JIA, HONG ZHANG, ZHULIN BEMBENEK, SCOTT DAMIAN SU, WEI-GUO JONES, WILLIAM MOORE |
| description | The invention relates to novel heteroaryl and heterocycle compounds of formula I and pharmaceutical compositions comprising them, uses and methods thereof for inhibiting the activity of PI3K and for treating inflammatory and autoimmune diseases and cancer.
La présente invention concerne de nouveaux composés hétéroaryliques et hétérocycliques de formule I et des compositions pharmaceutiques comprenant ceux-ci, leurs utilisations et procédés pour inhiber l'activité de la PI3K et traiter des maladies inflammatoires et auto-immunes ainsi que le cancer. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_WO2016119707A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>WO2016119707A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_WO2016119707A13</originalsourceid><addsrcrecordid>eNrjZHDx8w9z9VHwcA1xDfJ3DIr0UXD0c4FynSOdfVwVnP19A_xD_VyCdSDMYM8QT3-_YLA6X9cQD3-XYB4G1rTEnOJUXijNzaDs5hri7KGbWpAfn1pckJicmpdaEh_ub2RgaGZoaGluYO5oaEycKgAs2Sz-</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS</title><source>esp@cenet</source><creator>LEBSACK, ALEC DONALD ; ECCLES, WENDY ; DAI, GUANGXIU ; CHAI, WENYING ; MEDUNA, STEVEN PAUL ; KEITH, JOHN MATTHEW ; VENABLE, JENNIFER DIANE ; WENG, JIANYANG ; SMITH, RUSSELL CHRISTOPHER ; JIA, HONG ; ZHANG, ZHULIN ; BEMBENEK, SCOTT DAMIAN ; SU, WEI-GUO ; JONES, WILLIAM MOORE</creator><creatorcontrib>LEBSACK, ALEC DONALD ; ECCLES, WENDY ; DAI, GUANGXIU ; CHAI, WENYING ; MEDUNA, STEVEN PAUL ; KEITH, JOHN MATTHEW ; VENABLE, JENNIFER DIANE ; WENG, JIANYANG ; SMITH, RUSSELL CHRISTOPHER ; JIA, HONG ; ZHANG, ZHULIN ; BEMBENEK, SCOTT DAMIAN ; SU, WEI-GUO ; JONES, WILLIAM MOORE</creatorcontrib><description>The invention relates to novel heteroaryl and heterocycle compounds of formula I and pharmaceutical compositions comprising them, uses and methods thereof for inhibiting the activity of PI3K and for treating inflammatory and autoimmune diseases and cancer.
La présente invention concerne de nouveaux composés hétéroaryliques et hétérocycliques de formule I et des compositions pharmaceutiques comprenant ceux-ci, leurs utilisations et procédés pour inhiber l'activité de la PI3K et traiter des maladies inflammatoires et auto-immunes ainsi que le cancer.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2016</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160804&DB=EPODOC&CC=WO&NR=2016119707A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76516</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160804&DB=EPODOC&CC=WO&NR=2016119707A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>LEBSACK, ALEC DONALD</creatorcontrib><creatorcontrib>ECCLES, WENDY</creatorcontrib><creatorcontrib>DAI, GUANGXIU</creatorcontrib><creatorcontrib>CHAI, WENYING</creatorcontrib><creatorcontrib>MEDUNA, STEVEN PAUL</creatorcontrib><creatorcontrib>KEITH, JOHN MATTHEW</creatorcontrib><creatorcontrib>VENABLE, JENNIFER DIANE</creatorcontrib><creatorcontrib>WENG, JIANYANG</creatorcontrib><creatorcontrib>SMITH, RUSSELL CHRISTOPHER</creatorcontrib><creatorcontrib>JIA, HONG</creatorcontrib><creatorcontrib>ZHANG, ZHULIN</creatorcontrib><creatorcontrib>BEMBENEK, SCOTT DAMIAN</creatorcontrib><creatorcontrib>SU, WEI-GUO</creatorcontrib><creatorcontrib>JONES, WILLIAM MOORE</creatorcontrib><title>NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS</title><description>The invention relates to novel heteroaryl and heterocycle compounds of formula I and pharmaceutical compositions comprising them, uses and methods thereof for inhibiting the activity of PI3K and for treating inflammatory and autoimmune diseases and cancer.
La présente invention concerne de nouveaux composés hétéroaryliques et hétérocycliques de formule I et des compositions pharmaceutiques comprenant ceux-ci, leurs utilisations et procédés pour inhiber l'activité de la PI3K et traiter des maladies inflammatoires et auto-immunes ainsi que le cancer.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2016</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZHDx8w9z9VHwcA1xDfJ3DIr0UXD0c4FynSOdfVwVnP19A_xD_VyCdSDMYM8QT3-_YLA6X9cQD3-XYB4G1rTEnOJUXijNzaDs5hri7KGbWpAfn1pckJicmpdaEh_ub2RgaGZoaGluYO5oaEycKgAs2Sz-</recordid><startdate>20160804</startdate><enddate>20160804</enddate><creator>LEBSACK, ALEC DONALD</creator><creator>ECCLES, WENDY</creator><creator>DAI, GUANGXIU</creator><creator>CHAI, WENYING</creator><creator>MEDUNA, STEVEN PAUL</creator><creator>KEITH, JOHN MATTHEW</creator><creator>VENABLE, JENNIFER DIANE</creator><creator>WENG, JIANYANG</creator><creator>SMITH, RUSSELL CHRISTOPHER</creator><creator>JIA, HONG</creator><creator>ZHANG, ZHULIN</creator><creator>BEMBENEK, SCOTT DAMIAN</creator><creator>SU, WEI-GUO</creator><creator>JONES, WILLIAM MOORE</creator><scope>EVB</scope></search><sort><creationdate>20160804</creationdate><title>NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS</title><author>LEBSACK, ALEC DONALD ; ECCLES, WENDY ; DAI, GUANGXIU ; CHAI, WENYING ; MEDUNA, STEVEN PAUL ; KEITH, JOHN MATTHEW ; VENABLE, JENNIFER DIANE ; WENG, JIANYANG ; SMITH, RUSSELL CHRISTOPHER ; JIA, HONG ; ZHANG, ZHULIN ; BEMBENEK, SCOTT DAMIAN ; SU, WEI-GUO ; JONES, WILLIAM MOORE</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_WO2016119707A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2016</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>LEBSACK, ALEC DONALD</creatorcontrib><creatorcontrib>ECCLES, WENDY</creatorcontrib><creatorcontrib>DAI, GUANGXIU</creatorcontrib><creatorcontrib>CHAI, WENYING</creatorcontrib><creatorcontrib>MEDUNA, STEVEN PAUL</creatorcontrib><creatorcontrib>KEITH, JOHN MATTHEW</creatorcontrib><creatorcontrib>VENABLE, JENNIFER DIANE</creatorcontrib><creatorcontrib>WENG, JIANYANG</creatorcontrib><creatorcontrib>SMITH, RUSSELL CHRISTOPHER</creatorcontrib><creatorcontrib>JIA, HONG</creatorcontrib><creatorcontrib>ZHANG, ZHULIN</creatorcontrib><creatorcontrib>BEMBENEK, SCOTT DAMIAN</creatorcontrib><creatorcontrib>SU, WEI-GUO</creatorcontrib><creatorcontrib>JONES, WILLIAM MOORE</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>LEBSACK, ALEC DONALD</au><au>ECCLES, WENDY</au><au>DAI, GUANGXIU</au><au>CHAI, WENYING</au><au>MEDUNA, STEVEN PAUL</au><au>KEITH, JOHN MATTHEW</au><au>VENABLE, JENNIFER DIANE</au><au>WENG, JIANYANG</au><au>SMITH, RUSSELL CHRISTOPHER</au><au>JIA, HONG</au><au>ZHANG, ZHULIN</au><au>BEMBENEK, SCOTT DAMIAN</au><au>SU, WEI-GUO</au><au>JONES, WILLIAM MOORE</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS</title><date>2016-08-04</date><risdate>2016</risdate><abstract>The invention relates to novel heteroaryl and heterocycle compounds of formula I and pharmaceutical compositions comprising them, uses and methods thereof for inhibiting the activity of PI3K and for treating inflammatory and autoimmune diseases and cancer.
La présente invention concerne de nouveaux composés hétéroaryliques et hétérocycliques de formule I et des compositions pharmaceutiques comprenant ceux-ci, leurs utilisations et procédés pour inhiber l'activité de la PI3K et traiter des maladies inflammatoires et auto-immunes ainsi que le cancer.</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | eng ; fre |
| recordid | cdi_epo_espacenet_WO2016119707A1 |
| source | esp@cenet |
| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-14T12%3A53%3A40IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=LEBSACK,%20ALEC%20DONALD&rft.date=2016-08-04&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EWO2016119707A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |