1-(DIHYDRONAPHTHALENYL)PYRIDONES AS MELANIN-CONCENTRATING HORMONE RECEPTOR 1 ANTAGONISTS

Provided are 1-(dihydronaphthalenyl)pyridones which are antagonists at the melanin-concentrating hormone receptor 1 (MCHR1), pharmaceutical compositions containing them, processes for their preparation, and their use in therapy for the treatment of obesity and diabetes. L'invention concerne des...

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Hauptverfasser: QIN, DONGHUI, WU, CHENGDE, YUAN, JIANGXING, CHRISTENSEN, SIEG, YU, HAIYU, ZHANG, ZHILIU
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WU, CHENGDE
YUAN, JIANGXING
CHRISTENSEN, SIEG
YU, HAIYU
ZHANG, ZHILIU
description Provided are 1-(dihydronaphthalenyl)pyridones which are antagonists at the melanin-concentrating hormone receptor 1 (MCHR1), pharmaceutical compositions containing them, processes for their preparation, and their use in therapy for the treatment of obesity and diabetes. L'invention concerne des 1-(dihydronaphtalényl)pyridones qui sont des antagonistes du récepteur 1 de l'hormone de concentration de la mélanine (MCHR1), des compositions pharmaceutiques les contenant, des procédés pour leur préparation et leur utilisation dans une thérapie pour le traitement de l'obésité et du diabète.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title 1-(DIHYDRONAPHTHALENYL)PYRIDONES AS MELANIN-CONCENTRATING HORMONE RECEPTOR 1 ANTAGONISTS
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