INDOLE DERIVATIVE MODULATORS OF THE ALPHA 7 NACHR

This invention relates to modulation of the a7 nicotinic acetylcholine receptor (nAChR) by a compound of formula (I) or a salt thereof: wherein R1 is imidazolyl, pyridinyl or pyrimidinyl, any of which is optionally substituted by one group independently selected from C1-3alkyl and C1-3alkoxy. Cette...

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creator DINNELL, KEVIN
description This invention relates to modulation of the a7 nicotinic acetylcholine receptor (nAChR) by a compound of formula (I) or a salt thereof: wherein R1 is imidazolyl, pyridinyl or pyrimidinyl, any of which is optionally substituted by one group independently selected from C1-3alkyl and C1-3alkoxy. Cette invention porte sur la modulation du récepteur nicotinique a7 de l'acétylcholine (nAChR) par un composé de formule (I) ou un sel de celui-ci : où R1 est imidazolyle, pyridinyle ou pyrimidinyle, n'importe lequel d'entre eux étant facultativement substitué par un groupe indépendamment choisi parmi alkyle en C1-3 et alcoxy en C1-3.
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Cette invention porte sur la modulation du récepteur nicotinique a7 de l'acétylcholine (nAChR) par un composé de formule (I) ou un sel de celui-ci : où R1 est imidazolyle, pyridinyle ou pyrimidinyle, n'importe lequel d'entre eux étant facultativement substitué par un groupe indépendamment choisi parmi alkyle en C1-3 et alcoxy en C1-3.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2010</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20101021&amp;DB=EPODOC&amp;CC=WO&amp;NR=2010119078A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76289</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&amp;date=20101021&amp;DB=EPODOC&amp;CC=WO&amp;NR=2010119078A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>DINNELL, KEVIN</creatorcontrib><title>INDOLE DERIVATIVE MODULATORS OF THE ALPHA 7 NACHR</title><description>This invention relates to modulation of the a7 nicotinic acetylcholine receptor (nAChR) by a compound of formula (I) or a salt thereof: wherein R1 is imidazolyl, pyridinyl or pyrimidinyl, any of which is optionally substituted by one group independently selected from C1-3alkyl and C1-3alkoxy. 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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title INDOLE DERIVATIVE MODULATORS OF THE ALPHA 7 NACHR
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