INTERMEDIATES AND PROCESSES FOR THE PREPARATION OF FLUOROGLYCOSIDE DERIVATIVES

The present invention provides processes for producing (2S,3R,4R,5S,6R)-5-fluoro-6- hydroxymethyl-2-[4-(4-methoxy-benzyl)-5-trifluoromethyl-1H-pyrazol-3-yloxy]- tetrahydro-pyran-3,4-diol or a tautomer or hydrate thereof, of high purity and in a relatively high yield suitable for use on an industrial...

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Hauptverfasser: GILL, HARPAL S, LEE, GEORGE E, POWERS, MATTHEW R, WEIBERTH, FRANZ J, ZHANG, JIUQING, PLETTENBURG, OLIVER, ROSSEN, KAI, GESSLER, SIMON, YU, YONG, PODESCHWA, MICHAEL, VANASSE, BENOIT J, SHRIMP, II, FREDERICK L, SUBOTKOWSKI, WITOLD, WEHLAN, HERMUT A
Format: Patent
Sprache:eng ; fre
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