PROCESS FOR PREPARATION OF (S) (N-[[3-[3-FLUORO-4-(4-MORPHOLINYL) HEN L -2-OXO-5-OXAZOLIDIN L METHYL]ACETAMIDE
The present invention provides novel process for preparation of (S)-N-[[3-[3-Fluoro-4-(4- morpholinyl)phenyl]-2-oxo-5-oxazolidinyl] methyl] -acetamide which comprises combining (R)-N-[3-[3-fluoro-4-morpholinyl phenyl]-2-oxo-5-oxazolidinyl]methylazide in suitable solvent, acetylating agent and acid i...
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Format: | Patent |
Sprache: | eng ; fre |
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Zusammenfassung: | The present invention provides novel process for preparation of (S)-N-[[3-[3-Fluoro-4-(4- morpholinyl)phenyl]-2-oxo-5-oxazolidinyl] methyl] -acetamide which comprises combining (R)-N-[3-[3-fluoro-4-morpholinyl phenyl]-2-oxo-5-oxazolidinyl]methylazide in suitable solvent, acetylating agent and acid in presence of a catalyst.
La présente invention concerne un nouveau processus de préparation de (S)-N-[[3-[3-Fluoro-4-(4- morpholinyl)phényl]-2-oxo-5-oxazolidinyle] méthyl] -acétamide qui consiste à combiner (R)-N-[3-[3-fluoro-4-morpholinyle phényl]-2-oxo-5-oxazolidinyl]méthylazide dans un solvant adapté, un agent d'acétylation et un acide en présence d'un catalyseur. |
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