BENZOXAZINONE AND BENZOXAZEPINONE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS

The present invention provides a compound of formula (I) wherein X is a structure of the following formula (i), (ii), (iii), or iv G is O, or S; U is -(CR3R4)n-; W is CH2NHC(=G)R1, CH2NH-het, CH2-G-het, CH2het, C(=O)NHR2; and Y1, Y2 and Y3 are independently CH, or CF. The compounds of the present in...

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Bibliographische Detailangaben
Hauptverfasser:	RENSLO, ADAM, ROBERT, LUEHR, GARY, WAYNE, GAO, HONGWU, VENKATA NAGENDRA JOSYULA, VARA, PRASAD, GORDEEV, MIKHAIL
Format:	Patent
Sprache:	eng ; fre
Schlagworte:	CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:	The present invention provides a compound of formula (I) wherein X is a structure of the following formula (i), (ii), (iii), or iv G is O, or S; U is -(CR3R4)n-; W is CH2NHC(=G)R1, CH2NH-het, CH2-G-het, CH2het, C(=O)NHR2; and Y1, Y2 and Y3 are independently CH, or CF. The compounds of the present invention are useful as antibacterial agents. La présente invention concerne un composé de formule I où X représente une structure de formule i, ii, iii ou iv suivante; G représente O ou S; U représente -(CR3R4)n-; W représente CH2NHC(=G)R1, CH2NH-het, CH2-G-het, CH2het, C(=O)NHR2; et Y1, Y2 et Y3 représentent chacun indépendamment CH ou CF. Les composés selon la présente invention peuvent être employés en tant qu'agents antibactériens.