PROCESSES FOR PREPARING 4-(PHENOXY-5-METHYL-PYRIMIDIN-4-YLOXY)PIPERIDINE-1-CARBOXYLIC ACID DERIVATIVES AND RELATED COMPOUNDS

PROCESSES FOR PREPARING 4-(PHENOXY-5-METHYL-PYRIMIDIN-4-YLOXY)PIPERIDINE-1-CARBOXYLIC ACID DERIVATIVES AND RELATED COMPOUNDS

The invention discloses: A process for preparing a compound of Formula (I); wherein said process comprises reacting a compound of Formula (II); wherein L2 is a leaving group, with compound of Formula (III) in the presence of a base and a salt, thereby forming the compound of Formula (I). The substit...

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Bibliographische Detailangaben
Hauptverfasser: GHARBAOUI, TAWFIK, KATO, NAOMI, S, KRISHNAN, ASHWIN, M, THROOP, BEVERLY, WOLGAST, FRITCH, JOHN, R
Format: Patent
Sprache:eng ; fre
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Beschreibung
Zusammenfassung:The invention discloses: A process for preparing a compound of Formula (I); wherein said process comprises reacting a compound of Formula (II); wherein L2 is a leaving group, with compound of Formula (III) in the presence of a base and a salt, thereby forming the compound of Formula (I). The substituents and variables are defined in the claims. L'invention concerne un procédé d'élaboration de composé de formule (I) : réaction entre un composé de formule (II), L2 étant un groupe partant, et un composé de formule (III), en présence d'une base et d'un sel, ce qui donne le composé de formule (I). Les revendications de brevet définissent les substituants et les variables propres à l'invention.