PROCESS FOR THE PREPARATION OF (2S)-3-[4-({[4-(AMINOCARBONYL)-1-PIPERIDINYL]CARBONYL}OXY) PHENYL]2-{((2S)-4-METHYL-2-{[2-(2-METHYLPHENOXY)ACETYL]AMINO}PENTANOYL)AMINO[PROPANOIC ACID AND INTERMEDIATES THEREFORE

The present invention relates to a new process for preparing a compound (I) known in the art as an 4-integrin antagonist, intermediates useful in the process, and to a process for the preparation of such intermediates. The present invention relates to a new process for preparing a compound (I) known...

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Bibliographische Detailangaben
Hauptverfasser: ADAMS, JOSEPH, PAUL, ANSON, MICHAEL, SIMON, GOODING, STEVE
Format: Patent
Sprache:eng ; fre
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Zusammenfassung:The present invention relates to a new process for preparing a compound (I) known in the art as an 4-integrin antagonist, intermediates useful in the process, and to a process for the preparation of such intermediates. The present invention relates to a new process for preparing a compound (I) known in the art as an alpha4-integrin antagonist, intermediates useful in the process, and to a process for the preparation of such intermediates. La présente invention concerne un nouveau procédé de préparation d'un composé (I) connu comme antagoniste de l'intégrine alpha 4, des intermédiaires utiles dans ledit procédé et un procédé de préparation desdits intermédiaires.