CRYSTALLIZED GLUCOCORTICOID RECEPTOR LIGAND BINDING DOMAIN POLYPEPTIDE AND SCREENING METHODS EMPLOYING SAME

A method of modifying a test nuclear receptor (NR) polypeptide is disclosed. The method provides a test NR polypeptide sequence having a characteristic that is targeted for modification; aligning the test NR polypeptide sequence with at least one reference NR polypeptide sequence for which an X-ray...

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Hauptverfasser: LAMBERT, MILLARD, H., III, DELVES, CHRISTOPHER, J, PEARCE, KENNETH, H, MONTANA, VALERIE, GAIL, BLEDSOE, RANDY, K, MCKEE, DAVID, D, XU, HUAQIANG, ERIC, APOLITO, CHRISTOPHER, J, STANLEY, THOMAS, B
Format: Patent
Sprache:eng ; fre
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