PROCESSES FOR PREPARING TRIAZOLE GLYCOLATE OXIDASE INHIBITORS

PROCESSES FOR PREPARING TRIAZOLE GLYCOLATE OXIDASE INHIBITORS

The present disclosure provides processes for preparing 1,2,3-tri-azole-4-carboxylic acid related compounds of formulae (I) and (II) via a Suzuki coupling reaction. The Suzuki coupling reaction is achieved by coupling a compound of formula (IV), a boron-containing derivative of 1,2,3-triazole-4-carb...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: CHAND, Pooran, CHOUDHARY, Sunil Kumar, FERNANDES, Miguel Xavier, MAAG, Hans, AKBARIROMANI, Elham, REVU, Omkar, SHEKHAWAT, Pavan, LEBLANC, Yves
Format: Patent
Sprache:eng
Schlagworte:
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Beschreibung
Zusammenfassung:The present disclosure provides processes for preparing 1,2,3-tri-azole-4-carboxylic acid related compounds of formulae (I) and (II) via a Suzuki coupling reaction. The Suzuki coupling reaction is achieved by coupling a compound of formula (IV), a boron-containing derivative of 1,2,3-triazole-4-carb oxylate, with a cycloalkyl phenyl halide or sulfonate of formula (V).