Processes for preparing a diazabicyclooctane compound

A process for preparing a diazabicyclooctane compound represented by the following formula (I):wherein A represents RcO-; B represents NH or NC1-6 alkyl; C represents a benzyl group; Rc represents a C1-6 alkyl group; A is substituted with one substituent Fn1, wherein Fn1 represents an azetidine grou...

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Bibliographische Detailangaben
Hauptverfasser: Sakamaki, Yoshiaki, Furuuchi, Takeshi, Abe, Takao
Format: Patent
Sprache:eng
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Zusammenfassung:A process for preparing a diazabicyclooctane compound represented by the following formula (I):wherein A represents RcO-; B represents NH or NC1-6 alkyl; C represents a benzyl group; Rc represents a C1-6 alkyl group; A is substituted with one substituent Fn1, wherein Fn1 represents an azetidine group; the process including: (a) silylating the compound represented by the following formula (IV-c):wherein in the formula (IV-c), OBn represents benzyloxy, and (b) carrying out an intramolecular urea formation reaction.