Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same

Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same

The present invention relates to novel mesylate salt of N-(5-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yppyrimidine-2-ylamino)-4-methoxy-2-morpholinophenyl)acrylamide, a novel crystalline form thereof, and a process for preparing the same. More specifically, the present invention relates t...

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Hauptverfasser: Oh, Se-Woong, Kim, Kyeong Bae, Oh, Sang Ho, Shin, Woo Seob, Ju, Hyun, Kim, Dong Kyun, Kim, Jong Gyun, Park, Su Min, Han, Tae Dong, Lee, Young Sung, Kang, Jeong Ki, Chung, Soo Yong, Lee, Seong Ran
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ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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creator Oh, Se-Woong
Kim, Kyeong Bae
Oh, Sang Ho
Shin, Woo Seob
Ju, Hyun
Kim, Dong Kyun
Kim, Jong Gyun
Park, Su Min
Han, Tae Dong
Lee, Young Sung
Kang, Jeong Ki
Chung, Soo Yong
Lee, Seong Ran
description The present invention relates to novel mesylate salt of N-(5-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yppyrimidine-2-ylamino)-4-methoxy-2-morpholinophenyl)acrylamide, a novel crystalline form thereof, and a process for preparing the same. More specifically, the present invention relates to mesylate salt of N-(5-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yl)pyrimidine-2-ylamino)-4-methoxy-2-morpholinophenyl)acrylamide, which is excellent in stability, solubility, and bioavailability when it is administered not only alone but also in combination with other drugs and which has a high purity, a crystalline form thereof, and a process for preparing the same.
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subjects ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
title Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same
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