Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same

Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same

The present invention relates to novel mesylate salt of N-(5-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yppyrimidine-2-ylamino)-4-methoxy-2-morpholinophenyl)acrylamide, a novel crystalline form thereof, and a process for preparing the same. More specifically, the present invention relates t...

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Bibliographische Detailangaben
Hauptverfasser: Oh, Se-Woong, Kim, Kyeong Bae, Oh, Sang Ho, Shin, Woo Seob, Ju, Hyun, Kim, Dong Kyun, Kim, Jong Gyun, Park, Su Min, Han, Tae Dong, Lee, Young Sung, Kang, Jeong Ki, Chung, Soo Yong, Lee, Seong Ran
Format: Patent
Sprache:eng
Schlagworte:
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
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Beschreibung
Zusammenfassung:The present invention relates to novel mesylate salt of N-(5-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yppyrimidine-2-ylamino)-4-methoxy-2-morpholinophenyl)acrylamide, a novel crystalline form thereof, and a process for preparing the same. More specifically, the present invention relates to mesylate salt of N-(5-(4-(4-((dimethylamino)methyl)-3-phenyl-1H-pyrazol-1-yl)pyrimidine-2-ylamino)-4-methoxy-2-morpholinophenyl)acrylamide, which is excellent in stability, solubility, and bioavailability when it is administered not only alone but also in combination with other drugs and which has a high purity, a crystalline form thereof, and a process for preparing the same.