Carboxamide derivative and its diastereomers in stable crystalline form
The present disclosure relates to solid crystalline forms of N-((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)-propan-2-yl)-5-(1-hydroxyethyl)-1H-pyrazole-3- carboxamide (I) and the diastereomers thereof, and to methods for preparing such crystalline forms. Compound (I)and the diastereomers ther...
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| creator | Heikkinen, Terhi Törmäkangas, Olli |
| description | The present disclosure relates to solid crystalline forms of N-((S)-1-(3-(3-chloro-4-cyanophenyl)-1H-pyrazol-1-yl)-propan-2-yl)-5-(1-hydroxyethyl)-1H-pyrazole-3- carboxamide (I) and the diastereomers thereof, and to methods for preparing such crystalline forms. Compound (I)and the diastereomers thereof are potent androgen receptor (AR) modulators useful as a medicament. |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES |
| title | Carboxamide derivative and its diastereomers in stable crystalline form |
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