POLYCYCLIC INDAZOLE-DERIVATIVES AND THEIR APPLICATION AS ERK INHIBITORS FOR CANCER TREATMENT
FIELD: medicine, pharmaceutics.SUBSTANCE: invention relates to particular compounds, which demonstrate inhibiting activity with respect to ERK, whose structure formula is given in description, to their pharmaceutically acceptable salts, based on them pharmaceutical composition and their application...
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| creator | DESAI JAGDISH PALIUOL SANIL PATEL MEKHAL SHIKH NENG-JANG SHIPPS DZHERAL'D V. ML TSUI KHONUNG ALKHASSAN ABDUL-BASIT ZHU KHUG KELLI DZHOZEF BOGA SOBKHANA BABU ZHU LIANG DOLL RONAL'D VANG DZHEJMS NAN JANG DENG JONGKI KUPER ALAN GAO KSJAOLEJ |
| description | FIELD: medicine, pharmaceutics.SUBSTANCE: invention relates to particular compounds, which demonstrate inhibiting activity with respect to ERK, whose structure formula is given in description, to their pharmaceutically acceptable salts, based on them pharmaceutical composition and their application for treatment of cancer, mediated by ERK activity.EFFECT: obtaining compounds, which demonstrate inhibiting activity with respect to ERK.5 cl
Изобретение относится к конкретным соединениям, проявляющим ингибирующую активность в отношении ERK, структурная формула которых указана в описании, их фармацевтически приемлемым солям, фармацевтической композиции на их основе и их применению для лечения рака, опосредованного активностью ERK. 5 н.п. ф-лы. |
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Изобретение относится к конкретным соединениям, проявляющим ингибирующую активность в отношении ERK, структурная формула которых указана в описании, их фармацевтически приемлемым солям, фармацевтической композиции на их основе и их применению для лечения рака, опосредованного активностью ERK. 5 н.п. ф-лы.</description><language>eng ; rus</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2013</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20130220&DB=EPODOC&CC=RU&NR=2475484C2$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20130220&DB=EPODOC&CC=RU&NR=2475484C2$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>DESAI JAGDISH</creatorcontrib><creatorcontrib>PALIUOL SANIL</creatorcontrib><creatorcontrib>PATEL MEKHAL</creatorcontrib><creatorcontrib>SHIKH NENG-JANG</creatorcontrib><creatorcontrib>SHIPPS DZHERAL'D V. ML</creatorcontrib><creatorcontrib>TSUI KHONUNG</creatorcontrib><creatorcontrib>ALKHASSAN ABDUL-BASIT</creatorcontrib><creatorcontrib>ZHU KHUG</creatorcontrib><creatorcontrib>KELLI DZHOZEF</creatorcontrib><creatorcontrib>BOGA SOBKHANA BABU</creatorcontrib><creatorcontrib>ZHU LIANG</creatorcontrib><creatorcontrib>DOLL RONAL'D</creatorcontrib><creatorcontrib>VANG DZHEJMS</creatorcontrib><creatorcontrib>NAN JANG</creatorcontrib><creatorcontrib>DENG JONGKI</creatorcontrib><creatorcontrib>KUPER ALAN</creatorcontrib><creatorcontrib>GAO KSJAOLEJ</creatorcontrib><title>POLYCYCLIC INDAZOLE-DERIVATIVES AND THEIR APPLICATION AS ERK INHIBITORS FOR CANCER TREATMENT</title><description>FIELD: medicine, pharmaceutics.SUBSTANCE: invention relates to particular compounds, which demonstrate inhibiting activity with respect to ERK, whose structure formula is given in description, to their pharmaceutically acceptable salts, based on them pharmaceutical composition and their application for treatment of cancer, mediated by ERK activity.EFFECT: obtaining compounds, which demonstrate inhibiting activity with respect to ERK.5 cl
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | POLYCYCLIC INDAZOLE-DERIVATIVES AND THEIR APPLICATION AS ERK INHIBITORS FOR CANCER TREATMENT |
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