AMINO DERIVATIVES OF THIAZOLE OR STEREOISOMERS THEREOF OR ADDITIVE SALTS THEREOF, METHODS FOR THEIR PRODUCTION, PHARMACEUTICAL COMPOSITIONS POSSESSING ACTIVITY IN RESPECT WITH CORTICOTROPIC HORMONE (CRF)

FIELD: chemistry of heterocyclic compounds; production of pharmaceutical compositions. SUBSTANCE: amino derivative of thiazole have formula I where R1 is H or C1-C5-alkyl; R2 is radical having formula A, B, or C ; R3 is C1-C5-alkyl, hydroxy C1-C5-alkyl, tetrahydropyrane-2yloxyalkyl or C3-C11-acyloxy...

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Hauptverfasser:	DANIEL' ANN ZHANN GJULLI, ZHIJ VIKTOR KARLOS KURTEMANSH, KLODI SJUZANN IVETT GOT'E, KAMIJ-ZHORZH VERMJUT, P'ER MARI AL'BERT ROZHE, MISHEL' ZHAKK ANRI ZHESLEN
Format:	Patent
Sprache:	eng
Schlagworte:	CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Zusammenfassung:	FIELD: chemistry of heterocyclic compounds; production of pharmaceutical compositions. SUBSTANCE: amino derivative of thiazole have formula I where R1 is H or C1-C5-alkyl; R2 is radical having formula A, B, or C ; R3 is C1-C5-alkyl, hydroxy C1-C5-alkyl, tetrahydropyrane-2yloxyalkyl or C3-C11-acyloxyalkyl, R4 is C3-C6-cycloalkyl, hydroxy C1-C5-alkyl, C2-C10-alkoxyalkyl, C- C11-cycloalkyloxyalkyl, hydroxyalkyl oxyalkyl C2-C10, alkoxyalkyl oxyalkyl C3-C12, acyloxyalkyl C3-C11 or alkyl thioalkyl C2-C10, R5 is C3-C6-cycloalkyl, optionally substituted phenyl, thienyl, pyridyl or radical having formula where R6-R14 are mentioned in claim 1. EFFECT: improved quality. 12 cl, 8 tbl