NOVEL BENZAMIDE DERIVATIVES
THE PRESENT INVENTION PROVIDES A NOVEL BENZAMIDE DERIVATIVE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, A METHOD FOR PREPARING THE SAME, AND A 5-HT4 RECEPTOR AGONIST CONTAINING THE SAME AS AN ACTIVE INGREDIENT. BENZAMIDE DERIVATIVES OF THE PRESENT INVENTION HAVE A SUPERIOR AFFINITY FOR 5-HT4 RECE...
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Format: | Patent |
Sprache: | eng |
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Zusammenfassung: | THE PRESENT INVENTION PROVIDES A NOVEL BENZAMIDE DERIVATIVE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, A METHOD FOR PREPARING THE SAME, AND A 5-HT4 RECEPTOR AGONIST CONTAINING THE SAME AS AN ACTIVE INGREDIENT. BENZAMIDE DERIVATIVES OF THE PRESENT INVENTION HAVE A SUPERIOR AFFINITY FOR 5-HT4 RECEPTORS, A CAPABILITY TO REDUCE A GASTRIC EMPTYING TIME AND A LOW TOXICITY, AND CONSEQUENTLY ARE THERAPEUTICALLY EFFECTIVE FOR THE TREATMENT OF A VARIETY OF DISEASES ASSOCIATED WITH 5-HT4 RECEPTORS. |
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