NOVEL BENZAMIDE DERIVATIVES

THE PRESENT INVENTION PROVIDES A NOVEL BENZAMIDE DERIVATIVE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, A METHOD FOR PREPARING THE SAME, AND A 5-HT4 RECEPTOR AGONIST CONTAINING THE SAME AS AN ACTIVE INGREDIENT. BENZAMIDE DERIVATIVES OF THE PRESENT INVENTION HAVE A SUPERIOR AFFINITY FOR 5-HT4 RECE...

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Hauptverfasser: SOHN, JU-HEE, CHOI, SUNG-HAK, KIM, MI-YEON, KIM, SOON-HOE, IM, WEON-BIN, CHOI, SUN-HO, SUNG, HYUN-JUNG, SOHN, TAE-KYOUNG, CHO, KANG-HUN
Format: Patent
Sprache:eng
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Zusammenfassung:THE PRESENT INVENTION PROVIDES A NOVEL BENZAMIDE DERIVATIVE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, A METHOD FOR PREPARING THE SAME, AND A 5-HT4 RECEPTOR AGONIST CONTAINING THE SAME AS AN ACTIVE INGREDIENT. BENZAMIDE DERIVATIVES OF THE PRESENT INVENTION HAVE A SUPERIOR AFFINITY FOR 5-HT4 RECEPTORS, A CAPABILITY TO REDUCE A GASTRIC EMPTYING TIME AND A LOW TOXICITY, AND CONSEQUENTLY ARE THERAPEUTICALLY EFFECTIVE FOR THE TREATMENT OF A VARIETY OF DISEASES ASSOCIATED WITH 5-HT4 RECEPTORS.