MACROCYCLIC CARBOXYLIC ACIDS AND ACYLSULFONAMIDES AS INHIBITORS OF HCV REPLICATION

THE PRESENT INVENTION PROVIDES COMPOUNDS OF THE GENERAL FORMULAS I-IX, AS WELL AS COMPOSITIONS, INCLUDING PHARMACEUTICAL COMPOSITIONS, COMPRISING A SUBJECT COMPOUND. THE PRESENT INVENTION FURTHER PROVIDES TREATMENT METHODS, INCLUDING METHODS OF TREATING A HEPATITIS C VIRUS INFECTION AND METHODS OF T...

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Hauptverfasser: ANDREWS, STEVEN WADE, KENNEDY, APRIL LAYNE, WOODARD, BENJAMIN T, WENGLOSKY, STEVEN MARK, JIANG, YUTONG, MADDURU, MACHENDER R, JOSEY, JOHN ANTHONY, SCOTT D. SEIWERT, DOHERTY, GEORGE ANDREW, CONDROWSKI, KEVIN RONALD, BLATT, LAWRENCE M, STENGEL, PETER JOHN
Format: Patent
Sprache:eng
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Zusammenfassung:THE PRESENT INVENTION PROVIDES COMPOUNDS OF THE GENERAL FORMULAS I-IX, AS WELL AS COMPOSITIONS, INCLUDING PHARMACEUTICAL COMPOSITIONS, COMPRISING A SUBJECT COMPOUND. THE PRESENT INVENTION FURTHER PROVIDES TREATMENT METHODS, INCLUDING METHODS OF TREATING A HEPATITIS C VIRUS INFECTION AND METHODS OF TREATING LIVER FIBROSIS, THE METHODS GENERALLY INVOLVING ADMINISTERING TO AN INDIVIDUAL IN NEED THEREOF AN EFFECTIVE AMOUNT OF A SUBJECT COMPOUND OR COMPOSITION.