METHODS OF MAKING HIV-PROTEASE INHIBITORS AND INTERMEDIATES FOR MAKING HIV-PROTEASE INHIBITORS

HIV PROTEASE INHIBITORS INHIBIT OR BLOCK THE BIOLOGICAL ACTIVITY OF THE HIV PROTEASE ENZYME, CAUSING THE REPLICATION OF THE HIV VIRUS TO TERMINATE. THESE COMPOUNDS CAN BE PREPARED BY THE NOVEL METHODS OF THE PRESENT INVENTION USING THE NOVEL INVENTIVE INTERMEDIATES.

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Hauptverfasser: JULIETTE K. BUSSE, KATHLEEN R. WHITTEN, KIM F. ALBIZATI, ROBERT J. SZENDROI, TRAVIS P. REMARCHUK, SRINIVASAN BABU, BENNETT C. BORER
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Sprache:eng
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Zusammenfassung:HIV PROTEASE INHIBITORS INHIBIT OR BLOCK THE BIOLOGICAL ACTIVITY OF THE HIV PROTEASE ENZYME, CAUSING THE REPLICATION OF THE HIV VIRUS TO TERMINATE. THESE COMPOUNDS CAN BE PREPARED BY THE NOVEL METHODS OF THE PRESENT INVENTION USING THE NOVEL INVENTIVE INTERMEDIATES.