PROCESS FOR PREPARING -CARBOXY BENZYL ACETOAMIDO PENICILLANIC SALTS
Title compds. I; M = Na, K, organic amine (H NR3), R = C2-5 alkyl) were prepd. by the reaction of 6-aminopenicillanic acid with anhydride(IV) in organic solvent. Thus, anhydride(IV) was prepd. by the reaction of acylhalide and synthetic intermediate(III) obtained from phenylmalonic acid with N, N...
Gespeichert in:
Hauptverfasser: | , |
---|---|
Format: | Patent |
Sprache: | eng |
Schlagworte: | |
Online-Zugang: | Volltext bestellen |
Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
Zusammenfassung: | Title compds. I; M = Na, K, organic amine (H NR3), R = C2-5 alkyl) were prepd. by the reaction of 6-aminopenicillanic acid with anhydride(IV) in organic solvent. Thus, anhydride(IV) was prepd. by the reaction of acylhalide and synthetic intermediate(III) obtained from phenylmalonic acid with N, N' -bistrialkylsilylimidazolidinone (II), and anhydride(IV), R1,R2,R3 are same or not, C1-3 alkyl, R4 - R5R6R7C or C2H5O-, R5,R6R7 are same or not, C1-3 alkyl) was reacted with 6-aminopenicillanic acid in organic solvent to give I. |
---|