THE FABRICATION METHOD OF INTERMEDIATE FOR FABRICATING EDOXABANE AND THE FABRICATION METHOD OF EDOXABANE

The present invention relates to a method for manufacturing intermediates for manufacturing edoxaban and a method for manufacturing edoxaban. More specifically, the present invention relates to: a method for manufacturing intermediates for manufacturing edoxaban which can obtain intermediates and ed...

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Bibliographische Detailangaben
Hauptverfasser: JAYAPRAKASH NEERASA, CHUNG HUN SUK
Format: Patent
Sprache:eng ; kor
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Beschreibung
Zusammenfassung:The present invention relates to a method for manufacturing intermediates for manufacturing edoxaban and a method for manufacturing edoxaban. More specifically, the present invention relates to: a method for manufacturing intermediates for manufacturing edoxaban which can obtain intermediates and edoxaban in high yield and purity without using EDCI and HOBt as reaction reagents; and a method for manufacturing edoxaban. 에독사반의 제조용 중간체의 제조 방법 및 에독사반의 제조 방법에 관한 것으로, EDCI와 HOBt를 반응 시약으로 사용하지 않으면서, 높은 수율과 순도로 에독사반의 제조용 중간체 및 에독사반을 얻을 수 있는 에독사반의 제조용 중간체의 제조 방법 및 에독사반의 제조 방법에 관한 것이다.