(2,3-D)THIENOPYRIMIDINE DERIVATIVE AND ITS SALT

NEW MATERIAL:The compound (salt) of formula I [R and R are H, halogen, 1-6C alkyl or R and R together form a 5-6-membered alkylene ring; R and R are H or 1-6C alkyl; R is H, 1-6C alkyl, group of formula II (m is 1-3; X is halogen), etc.; Ar is (substituted) phenyl, etc.; n is 2-3]. EXAMPLE:6-Methyl-...

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Hauptverfasser: KIKUMOTO RIYOUJI, EGAWA MITSUO, NITSUTA KAZUMASA, TOBE AKIHIRO, NINOMIYA KUNIHIRO
Format: Patent
Sprache:eng
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Zusammenfassung:NEW MATERIAL:The compound (salt) of formula I [R and R are H, halogen, 1-6C alkyl or R and R together form a 5-6-membered alkylene ring; R and R are H or 1-6C alkyl; R is H, 1-6C alkyl, group of formula II (m is 1-3; X is halogen), etc.; Ar is (substituted) phenyl, etc.; n is 2-3]. EXAMPLE:6-Methyl-4-phenyl-2-piperazinyl-[2,3-d]thienopyrimidine. USE:Psychopharmaceuticals. PREPARATION:The compound of formula I can be produced, e.g. by dissolving the 2-halo-6-substituted-4-phenyl-[2,3-d]thienopyrimidine of formula III (Y is halogen) in a solvent such as chloroform, and reacting with the piperazine compound of formula IV.