SUBSTITUTED 5H-PYRIMIDO(5,4-B)INDOLE, MANUFACTURE AND PSYCHOTIC MEDICINE
Substituted 5H-pyrimido[5,4-b]indoles of Formula I (I) wherein R2 is halogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; C1-5-alkyl, cycloalkyl, aralkyl, or aryl; ORI, SOnRI with n being 0, 1, or 2, or wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl...
Gespeichert in:
| Hauptverfasser: | , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | eng |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | ANDOREASU FUUTO HERUBERUTO HANSU SHIYUNAIDAA DEIITAA RAATSU BUORUFUGANGU KEERU RARUFU SHIYUMIIHIEN DEIITAA ZAIDERUMAN |
| description | Substituted 5H-pyrimido[5,4-b]indoles of Formula I (I) wherein R2 is halogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; C1-5-alkyl, cycloalkyl, aralkyl, or aryl; ORI, SOnRI with n being 0, 1, or 2, or wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, C3-5-alkenyl, cycloalkyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; and RA is hydrogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; halogen, nitro, ORI, SOnRI with n being 0, 1, or 2, wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, cycloalkyl, C3-5-alkenyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; or PO(OR)2 wherein R is C1-5-alkyl, exhibit strong affinity for binding to benzodiazepine receptors. The novel compounds are suitable for use in psychopharmaceutical preparations. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_JPS59130288A</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>JPS59130288A</sourcerecordid><originalsourceid>FETCH-epo_espacenet_JPS59130288A3</originalsourceid><addsrcrecordid>eNrjZPAIDnUKDvEMCQ1xdVEw9dANiAzy9PV08dcw1THRddL09HPx93HVUfB19At1c3QOCQ1yVXD0c1EICI509vAP8XRW8HV18XT29HPlYWBNS8wpTuWF0twMim6uIc4euqkF-fGpxQWJyal5qSXxXgHBppaGxgZGFhaOxsSoAQDsOizk</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>SUBSTITUTED 5H-PYRIMIDO(5,4-B)INDOLE, MANUFACTURE AND PSYCHOTIC MEDICINE</title><source>esp@cenet</source><creator>ANDOREASU FUUTO ; HERUBERUTO HANSU SHIYUNAIDAA ; DEIITAA RAATSU ; BUORUFUGANGU KEERU ; RARUFU SHIYUMIIHIEN ; DEIITAA ZAIDERUMAN</creator><creatorcontrib>ANDOREASU FUUTO ; HERUBERUTO HANSU SHIYUNAIDAA ; DEIITAA RAATSU ; BUORUFUGANGU KEERU ; RARUFU SHIYUMIIHIEN ; DEIITAA ZAIDERUMAN</creatorcontrib><description>Substituted 5H-pyrimido[5,4-b]indoles of Formula I (I) wherein R2 is halogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; C1-5-alkyl, cycloalkyl, aralkyl, or aryl; ORI, SOnRI with n being 0, 1, or 2, or wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, C3-5-alkenyl, cycloalkyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; and RA is hydrogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; halogen, nitro, ORI, SOnRI with n being 0, 1, or 2, wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, cycloalkyl, C3-5-alkenyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; or PO(OR)2 wherein R is C1-5-alkyl, exhibit strong affinity for binding to benzodiazepine receptors. The novel compounds are suitable for use in psychopharmaceutical preparations.</description><language>eng</language><subject>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>1984</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19840726&DB=EPODOC&CC=JP&NR=S59130288A$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76289</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19840726&DB=EPODOC&CC=JP&NR=S59130288A$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>ANDOREASU FUUTO</creatorcontrib><creatorcontrib>HERUBERUTO HANSU SHIYUNAIDAA</creatorcontrib><creatorcontrib>DEIITAA RAATSU</creatorcontrib><creatorcontrib>BUORUFUGANGU KEERU</creatorcontrib><creatorcontrib>RARUFU SHIYUMIIHIEN</creatorcontrib><creatorcontrib>DEIITAA ZAIDERUMAN</creatorcontrib><title>SUBSTITUTED 5H-PYRIMIDO(5,4-B)INDOLE, MANUFACTURE AND PSYCHOTIC MEDICINE</title><description>Substituted 5H-pyrimido[5,4-b]indoles of Formula I (I) wherein R2 is halogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; C1-5-alkyl, cycloalkyl, aralkyl, or aryl; ORI, SOnRI with n being 0, 1, or 2, or wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, C3-5-alkenyl, cycloalkyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; and RA is hydrogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; halogen, nitro, ORI, SOnRI with n being 0, 1, or 2, wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, cycloalkyl, C3-5-alkenyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; or PO(OR)2 wherein R is C1-5-alkyl, exhibit strong affinity for binding to benzodiazepine receptors. The novel compounds are suitable for use in psychopharmaceutical preparations.</description><subject>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>1984</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZPAIDnUKDvEMCQ1xdVEw9dANiAzy9PV08dcw1THRddL09HPx93HVUfB19At1c3QOCQ1yVXD0c1EICI509vAP8XRW8HV18XT29HPlYWBNS8wpTuWF0twMim6uIc4euqkF-fGpxQWJyal5qSXxXgHBppaGxgZGFhaOxsSoAQDsOizk</recordid><startdate>19840726</startdate><enddate>19840726</enddate><creator>ANDOREASU FUUTO</creator><creator>HERUBERUTO HANSU SHIYUNAIDAA</creator><creator>DEIITAA RAATSU</creator><creator>BUORUFUGANGU KEERU</creator><creator>RARUFU SHIYUMIIHIEN</creator><creator>DEIITAA ZAIDERUMAN</creator><scope>EVB</scope></search><sort><creationdate>19840726</creationdate><title>SUBSTITUTED 5H-PYRIMIDO(5,4-B)INDOLE, MANUFACTURE AND PSYCHOTIC MEDICINE</title><author>ANDOREASU FUUTO ; HERUBERUTO HANSU SHIYUNAIDAA ; DEIITAA RAATSU ; BUORUFUGANGU KEERU ; RARUFU SHIYUMIIHIEN ; DEIITAA ZAIDERUMAN</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_JPS59130288A3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>1984</creationdate><topic>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>ANDOREASU FUUTO</creatorcontrib><creatorcontrib>HERUBERUTO HANSU SHIYUNAIDAA</creatorcontrib><creatorcontrib>DEIITAA RAATSU</creatorcontrib><creatorcontrib>BUORUFUGANGU KEERU</creatorcontrib><creatorcontrib>RARUFU SHIYUMIIHIEN</creatorcontrib><creatorcontrib>DEIITAA ZAIDERUMAN</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>ANDOREASU FUUTO</au><au>HERUBERUTO HANSU SHIYUNAIDAA</au><au>DEIITAA RAATSU</au><au>BUORUFUGANGU KEERU</au><au>RARUFU SHIYUMIIHIEN</au><au>DEIITAA ZAIDERUMAN</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>SUBSTITUTED 5H-PYRIMIDO(5,4-B)INDOLE, MANUFACTURE AND PSYCHOTIC MEDICINE</title><date>1984-07-26</date><risdate>1984</risdate><abstract>Substituted 5H-pyrimido[5,4-b]indoles of Formula I (I) wherein R2 is halogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; C1-5-alkyl, cycloalkyl, aralkyl, or aryl; ORI, SOnRI with n being 0, 1, or 2, or wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, C3-5-alkenyl, cycloalkyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; and RA is hydrogen; the oxadiazolyl group wherein R'' is lower alkyl with up to 3 carbon atoms; halogen, nitro, ORI, SOnRI with n being 0, 1, or 2, wherein RI is hydrogen, C1-5-alkyl, cycloalkyl, aralkyl, or aryl; wherein RII and RIII are hydrogen, C1-5-alkyl, cycloalkyl, C3-5-alkenyl, aralkyl, aryl, or, with the connecting N-atom, a 5- or 6-membered heterocyclic ring; or PO(OR)2 wherein R is C1-5-alkyl, exhibit strong affinity for binding to benzodiazepine receptors. The novel compounds are suitable for use in psychopharmaceutical preparations.</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | eng |
| recordid | cdi_epo_espacenet_JPS59130288A |
| source | esp@cenet |
| subjects | ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | SUBSTITUTED 5H-PYRIMIDO(5,4-B)INDOLE, MANUFACTURE AND PSYCHOTIC MEDICINE |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-05T11%3A55%3A10IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=ANDOREASU%20FUUTO&rft.date=1984-07-26&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EJPS59130288A%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |