8-AMINO-PYRIDO(1,2,3-D,E)(1,3,4)BENZOXADIAZINE DERIVATIVE
8-Amino-pyrido(1,2,3-de)(1,3,4)benzoxadiazine derivs. of formula (I) and their enantiomers, hydrates and salts are new. A = amino or alkylamino; R1 = H or 1-3C alkyl opt. substd. by OH or halogen; R2 = H or Me; R3 = H or 1-4C alkyl; B = H; 1-4C alkyl opt. substd. by OH, OMe, NH2, NHMe or NMe2; or 5-...
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| creator | KAARUUGEORUKU METSUTSUGAA TOOMASU IECHIYU RAINAA ENDERUMAN UBE PEETAAZEN HAINTSUUGEORUKU BETSUTSUSHIYUTAIN KURAUSUUDEIITAA BUREMU MIHIYAERU SHIYUTEGEMAN MARUTEIN SHIEERU |
| description | 8-Amino-pyrido(1,2,3-de)(1,3,4)benzoxadiazine derivs. of formula (I) and their enantiomers, hydrates and salts are new. A = amino or alkylamino; R1 = H or 1-3C alkyl opt. substd. by OH or halogen; R2 = H or Me; R3 = H or 1-4C alkyl; B = H; 1-4C alkyl opt. substd. by OH, OMe, NH2, NHMe or NMe2; or 5-methyl-2-oxo-1,3- dioxol-4-ylmethyl; X1 = H or halogen; Z = a gp. of formula Z1-Z12. R4 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl or 1-3C acyl; R5 = H, Me, Ph, thienyl or pyridyl; R6-R8 = H or 1-4C alkyl; R9 = H, Me or CH2NR7R8; R10 = H, 1-4C alkyl, amino, opt. OH-substd. mono- or di(1-2C alkyl)amino, 1-4C aminoalkyl, (1-4C)alkylamino(1-4C)alkyl or 1-imidazolyl; R11=H, OH, OMe, SMe, halogen, Me or CH2OH; R12 = H or Me; R13-R15 = H or 1-4C alkyl. Also claimed are intermediates of formula (II). X2 = halogen. |
| format | Patent |
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A = amino or alkylamino; R1 = H or 1-3C alkyl opt. substd. by OH or halogen; R2 = H or Me; R3 = H or 1-4C alkyl; B = H; 1-4C alkyl opt. substd. by OH, OMe, NH2, NHMe or NMe2; or 5-methyl-2-oxo-1,3- dioxol-4-ylmethyl; X1 = H or halogen; Z = a gp. of formula Z1-Z12. R4 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl or 1-3C acyl; R5 = H, Me, Ph, thienyl or pyridyl; R6-R8 = H or 1-4C alkyl; R9 = H, Me or CH2NR7R8; R10 = H, 1-4C alkyl, amino, opt. OH-substd. mono- or di(1-2C alkyl)amino, 1-4C aminoalkyl, (1-4C)alkylamino(1-4C)alkyl or 1-imidazolyl; R11=H, OH, OMe, SMe, halogen, Me or CH2OH; R12 = H or Me; R13-R15 = H or 1-4C alkyl. Also claimed are intermediates of formula (II). X2 = halogen.</description><edition>6</edition><language>eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>1996</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19960227&DB=EPODOC&CC=JP&NR=H0853460A$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25543,76293</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19960227&DB=EPODOC&CC=JP&NR=H0853460A$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>KAARUUGEORUKU METSUTSUGAA</creatorcontrib><creatorcontrib>TOOMASU IECHIYU</creatorcontrib><creatorcontrib>RAINAA ENDERUMAN</creatorcontrib><creatorcontrib>UBE PEETAAZEN</creatorcontrib><creatorcontrib>HAINTSUUGEORUKU BETSUTSUSHIYUTAIN</creatorcontrib><creatorcontrib>KURAUSUUDEIITAA BUREMU</creatorcontrib><creatorcontrib>MIHIYAERU SHIYUTEGEMAN</creatorcontrib><creatorcontrib>MARUTEIN SHIEERU</creatorcontrib><title>8-AMINO-PYRIDO(1,2,3-D,E)(1,3,4)BENZOXADIAZINE DERIVATIVE</title><description>8-Amino-pyrido(1,2,3-de)(1,3,4)benzoxadiazine derivs. of formula (I) and their enantiomers, hydrates and salts are new. A = amino or alkylamino; R1 = H or 1-3C alkyl opt. substd. by OH or halogen; R2 = H or Me; R3 = H or 1-4C alkyl; B = H; 1-4C alkyl opt. substd. by OH, OMe, NH2, NHMe or NMe2; or 5-methyl-2-oxo-1,3- dioxol-4-ylmethyl; X1 = H or halogen; Z = a gp. of formula Z1-Z12. R4 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl or 1-3C acyl; R5 = H, Me, Ph, thienyl or pyridyl; R6-R8 = H or 1-4C alkyl; R9 = H, Me or CH2NR7R8; R10 = H, 1-4C alkyl, amino, opt. OH-substd. mono- or di(1-2C alkyl)amino, 1-4C aminoalkyl, (1-4C)alkylamino(1-4C)alkyl or 1-imidazolyl; R11=H, OH, OMe, SMe, halogen, Me or CH2OH; R12 = H or Me; R13-R15 = H or 1-4C alkyl. Also claimed are intermediates of formula (II). X2 = halogen.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>1996</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZLC00HX09fTz1w2IDPJ08dcw1DHSMdZ10XHVBDKNdUw0nVz9ovwjHF08HaM8_VwVXFyDPMMcQzzDXHkYWNMSc4pTeaE0N4OCm2uIs4duakF-fGpxQWJyal5qSbxXgIeBhamxiZmBozERSgCtuydh</recordid><startdate>19960227</startdate><enddate>19960227</enddate><creator>KAARUUGEORUKU METSUTSUGAA</creator><creator>TOOMASU IECHIYU</creator><creator>RAINAA ENDERUMAN</creator><creator>UBE PEETAAZEN</creator><creator>HAINTSUUGEORUKU BETSUTSUSHIYUTAIN</creator><creator>KURAUSUUDEIITAA BUREMU</creator><creator>MIHIYAERU SHIYUTEGEMAN</creator><creator>MARUTEIN SHIEERU</creator><scope>EVB</scope></search><sort><creationdate>19960227</creationdate><title>8-AMINO-PYRIDO(1,2,3-D,E)(1,3,4)BENZOXADIAZINE DERIVATIVE</title><author>KAARUUGEORUKU METSUTSUGAA ; TOOMASU IECHIYU ; RAINAA ENDERUMAN ; UBE PEETAAZEN ; HAINTSUUGEORUKU BETSUTSUSHIYUTAIN ; KURAUSUUDEIITAA BUREMU ; MIHIYAERU SHIYUTEGEMAN ; MARUTEIN SHIEERU</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_JPH0853460A3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>1996</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>KAARUUGEORUKU METSUTSUGAA</creatorcontrib><creatorcontrib>TOOMASU IECHIYU</creatorcontrib><creatorcontrib>RAINAA ENDERUMAN</creatorcontrib><creatorcontrib>UBE PEETAAZEN</creatorcontrib><creatorcontrib>HAINTSUUGEORUKU BETSUTSUSHIYUTAIN</creatorcontrib><creatorcontrib>KURAUSUUDEIITAA BUREMU</creatorcontrib><creatorcontrib>MIHIYAERU SHIYUTEGEMAN</creatorcontrib><creatorcontrib>MARUTEIN SHIEERU</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>KAARUUGEORUKU METSUTSUGAA</au><au>TOOMASU IECHIYU</au><au>RAINAA ENDERUMAN</au><au>UBE PEETAAZEN</au><au>HAINTSUUGEORUKU BETSUTSUSHIYUTAIN</au><au>KURAUSUUDEIITAA BUREMU</au><au>MIHIYAERU SHIYUTEGEMAN</au><au>MARUTEIN SHIEERU</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>8-AMINO-PYRIDO(1,2,3-D,E)(1,3,4)BENZOXADIAZINE DERIVATIVE</title><date>1996-02-27</date><risdate>1996</risdate><abstract>8-Amino-pyrido(1,2,3-de)(1,3,4)benzoxadiazine derivs. of formula (I) and their enantiomers, hydrates and salts are new. A = amino or alkylamino; R1 = H or 1-3C alkyl opt. substd. by OH or halogen; R2 = H or Me; R3 = H or 1-4C alkyl; B = H; 1-4C alkyl opt. substd. by OH, OMe, NH2, NHMe or NMe2; or 5-methyl-2-oxo-1,3- dioxol-4-ylmethyl; X1 = H or halogen; Z = a gp. of formula Z1-Z12. R4 = H, 1-4C alkyl (opt. substd. by OH or OMe), cyclopropyl or 1-3C acyl; R5 = H, Me, Ph, thienyl or pyridyl; R6-R8 = H or 1-4C alkyl; R9 = H, Me or CH2NR7R8; R10 = H, 1-4C alkyl, amino, opt. OH-substd. mono- or di(1-2C alkyl)amino, 1-4C aminoalkyl, (1-4C)alkylamino(1-4C)alkyl or 1-imidazolyl; R11=H, OH, OMe, SMe, halogen, Me or CH2OH; R12 = H or Me; R13-R15 = H or 1-4C alkyl. Also claimed are intermediates of formula (II). X2 = halogen.</abstract><edition>6</edition><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | 8-AMINO-PYRIDO(1,2,3-D,E)(1,3,4)BENZOXADIAZINE DERIVATIVE |
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