BENZOXAZEPINE COMPOUND

NEW MATERIAL:The compound of formula I {R and R are H or alkyl; R is H, alkyl or (substituted) phenylalkyl; R and R are H, halogen, alkyl, alkoxy, amino, etc.; X is NH; R is group of formula II (m is 0 or 1), formula III [R is alkyl, (substituted) phenylalkyl, etc.; R is H or alkoxy; n is 0 or 1], f...

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Hauptverfasser:	KUROITA TAKANOBU, FUKUDA TAKEMI, KAWAKITA TAKESHI, IKEZAWA RYUHEI
Format:	Patent
Sprache:	eng
Schlagworte:	CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:	NEW MATERIAL:The compound of formula I {R and R are H or alkyl; R is H, alkyl or (substituted) phenylalkyl; R and R are H, halogen, alkyl, alkoxy, amino, etc.; X is NH; R is group of formula II (m is 0 or 1), formula III [R is alkyl, (substituted) phenylalkyl, etc.; R is H or alkoxy; n is 0 or 1], formula IV [R is alkyl or (substituted) phenylalkyl; p and q are 0 or 1], etc.}. EXAMPLE:7-Chloro-5-methyl-N-(3-quinuclidinyl)-2,3,4,5-tetrahydro-1,5- benzoxazepine-9-carboxamide dihydrochloride. USE:A preventive and remedy for digestive diseases such as dyspepsia, delayed gastric emptying and peptic ulcer and remedy for emesis, central nervous system disorder, dementia, etc. PREPARATION:A carboxylic acid of formula V or its reactive derivative is made to react with a compound of formula R -XH.