N-(CYANOMETHYL)-4-(2-(4-MORPHOLINOPHENYLAMINO)PYRIMIDIN-4-YL) BENZAMIDE HYDROCHLORIDE

PROBLEM TO BE SOLVED: To provide stable novel salt forms of N-(cyanomethyl)-4-(2-(4-morpholinophenylamino) pyrimidin-4-yl) benzamide that are suitable for preparation of pharmaceutical formulations, and their therapeutic use.SOLUTION: The present invention relates to stable novel salt forms of N-(cy...

Ausführliche Beschreibung

Gespeichert in:
Bibliographische Detailangaben
Hauptverfasser: MATTHEW ROBERT WARR, YANG XING, JAMES ANDREW WHITNEY, BRANDON H BROWN, TROY REYNOLDS, SHI BIN, JEFFREY N HEMENWAY, ERNEST A CARRA, DEMITRIOS STEFANIDIS, WANG FANG, HENRY MORRISON
Format: Patent
Sprache:eng ; jpn
Schlagworte:
Online-Zugang:Volltext bestellen
Tags: Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
Beschreibung
Zusammenfassung:PROBLEM TO BE SOLVED: To provide stable novel salt forms of N-(cyanomethyl)-4-(2-(4-morpholinophenylamino) pyrimidin-4-yl) benzamide that are suitable for preparation of pharmaceutical formulations, and their therapeutic use.SOLUTION: The present invention relates to stable novel salt forms of N-(cyanomethyl)-4-(2-(4-morpholinophenylamino) pyrimidin-4-yl) benzamide and their therapeutic use, which are suitable for preparation of pharmaceutical formulations thereof.SELECTED DRAWING: Figure 1 【課題】医薬製剤の調製に適切である、安定した新規の塩形態のN−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミドおよびこれらの治療的使用を提供すること。【解決手段】本件発明は、安定である新規の塩の形態のN−(シアノメチル)−4−(2−(4−モルホリノフェニルアミノ)ピリミジン−4−イル)ベンズアミド、ならびに、これらの治療的使用に関するところのものであり、これは、その医薬製剤の調製に適切である。【選択図】 図1