SALTS OF HIV INHIBITOR COMPOUNDS
PROBLEM TO BE SOLVED: To provide salts of HIV inhibitor compounds.SOLUTION: The invention relates to salts of antiviral compounds, a composition containing such salts, a treatment method containing administration of such salts, a process and an intermediate useful for manufacturing such salts. The i...
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| creator | GRAETZ BENJAMIN R RICHARD P POLNIASZEK |
| description | PROBLEM TO BE SOLVED: To provide salts of HIV inhibitor compounds.SOLUTION: The invention relates to salts of antiviral compounds, a composition containing such salts, a treatment method containing administration of such salts, a process and an intermediate useful for manufacturing such salts. The invention provides stable salts of ethyl N-[(S)-({[(2R,5R)-5-(6-amino-9H-purine-9-yl)-4-fluoro-2,5-dihydrofuran-2-yl]oxy}methyl)phenoxyphosphinoyl]-L-alaninate which is physically more stable, easier to isolate and formulate than a free base type of the compound. |
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The invention provides stable salts of ethyl N-[(S)-({[(2R,5R)-5-(6-amino-9H-purine-9-yl)-4-fluoro-2,5-dihydrofuran-2-yl]oxy}methyl)phenoxyphosphinoyl]-L-alaninate which is physically more stable, easier to isolate and formulate than a free base type of the compound.</description><language>eng</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM ; CHEMISTRY ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2014</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20140703&DB=EPODOC&CC=JP&NR=2014122235A$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25543,76293</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20140703&DB=EPODOC&CC=JP&NR=2014122235A$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>GRAETZ BENJAMIN R</creatorcontrib><creatorcontrib>RICHARD P POLNIASZEK</creatorcontrib><title>SALTS OF HIV INHIBITOR COMPOUNDS</title><description>PROBLEM TO BE SOLVED: To provide salts of HIV inhibitor compounds.SOLUTION: The invention relates to salts of antiviral compounds, a composition containing such salts, a treatment method containing administration of such salts, a process and an intermediate useful for manufacturing such salts. 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| subjects | ACYCLIC OR CARBOCYCLIC COMPOUNDS ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM CHEMISTRY HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | SALTS OF HIV INHIBITOR COMPOUNDS |
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