AROMATIC DERIVATIVE AS HIV ASPARTYL PROTEASE INHIBITOR

PROBLEM TO BE SOLVED: To provide a new kind of compounds, and derivatives thereof permissible as pharmaceuticals. SOLUTION: There are provided HIV aspartyl protease inhibitors of the formula (I) and, when the compound of formula (I) contains an amino group, pharmaceutically acceptable ammonium salts...

Ausführliche Beschreibung

Gespeichert in:

Bibliographische Detailangaben
Hauptverfasser:	PERRON VALERIE, LAVALLEE JEAN-FRANCOIS, LEBERRE NICOLAS, STRANIX BRENT RICHARD
Format:	Patent
Sprache:	eng
Schlagworte:	ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
Online-Zugang:	Volltext bestellen
Tags:	Tag hinzufügen Keine Tags, Fügen Sie den ersten Tag hinzu!

Beschreibung
Zusammenfassung:	PROBLEM TO BE SOLVED: To provide a new kind of compounds, and derivatives thereof permissible as pharmaceuticals. SOLUTION: There are provided HIV aspartyl protease inhibitors of the formula (I) and, when the compound of formula (I) contains an amino group, pharmaceutically acceptable ammonium salts thereof, (wherein n is 3 or 4; R1may be, for example, iso-butyl; X and Y are same or different, and may be, for example, NH2and F; and R2and R3are as specifically defined herein). COPYRIGHT: (C)2010,JPO&INPIT