PROCEDIMENTO PER LA PREPARAZIONE DI EPIBATIDINA

The subject-matter of the invention is a process for preparing racemic or optically active epibatidine of formula which comprises cyclising a 1-ÄdiacylaminoÜ-2-Ä6'-chloro)-pyrid-3'-ylÜ-4-ÄaminoÜ-cyclohexane of general formula wherein Ac stands for an acyl group. The advantage of the proces...

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Hauptverfasser: TEMESVARI NATA MAJOR ESZTER, BLASKO GABOR, MANDI ATTILA, SZANTAY CSABA, SZALLAST TAMAS, LAX GYORGYI, FEKETE MARTON, SZANTAY CSABA JR, GIGLER GABOR, BALOGH NATA KARDOS ZSUZSANNA, SIMIG GYULA, DABRANT SANDOR, MOLDVAI ISTVAN
Format: Patent
Sprache:ita
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Zusammenfassung:The subject-matter of the invention is a process for preparing racemic or optically active epibatidine of formula which comprises cyclising a 1-ÄdiacylaminoÜ-2-Ä6'-chloro)-pyrid-3'-ylÜ-4-ÄaminoÜ-cyclohexane of general formula wherein Ac stands for an acyl group. The advantage of the process is that readily available starting materials are used and the procedure is suitable for industrial scale productions, too.